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Abarelix mai ƙarfi Gonadotropin-Sakin Hormone antagonist don Maganin Ciwon Prostate

Farashin: USD 100-200/g

  • Sunan samfur Abarelix
  • CAS No. 183552-38-7
  • MF Saukewa: C72H95ClN14O14
  • MW 1416.0631
  • EINECS 1592732-453-0
  • Yawan yawa 1.286
  • Wurin tafasa 1688.4°Cat760mmHg
  • Ma'anar walƙiya 974.9°C

Cikakken Bayani

Abarelix, wani decapeptide na roba, yana nuna babban aiki na gaba da gonadotropin-sakin hormone (GnRH). Ana amfani da shi da farko don kula da marasa lafiya da ke da ci-gaban ciwon daji na prostate waɗanda ba su dace da ƴan takara don luteinizing hormone-reaseing hormone agonists ko castration na tiyata ba. Ta hanyar hanawa kai tsaye na luteinizing hormone (LH) da kuma follicle-stimulating hormone (FSH), abarelix yadda ya kamata ya rage samar da testosterone daga ƙwanƙwasa. bari mu bincika alamun warkewa, hanyoyin aiki, da kuma amfani da abarelix.

Ana nuna Abarelix don maganin jin daɗi na marasa lafiya da ke fama da ciwon daji na prostate wanda ya dace da takamaiman sharuɗɗa. Ana ba da shawarar ga marasa lafiya waɗanda ba su dace da 'yan takara don agonists masu sakin hormone na luteinizing ba, sun ƙi simintin tiyata, kuma suna da ƙarin abubuwan haɗari kamar yuwuwar lalacewar jijiya saboda metastasis, urethra ko mafitsara ta hanyar toshewar ɓarna na gida ko metastasis, ko matsanancin ciwon ƙashi na ƙasusuwa da ke buƙatar ci gaba da jin zafi na narcotic.


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A matsayin injectable gonadotropin-releasing hormone antagonist (GnRH antagonist), abarelix yana taka muhimmiyar rawa wajen rage samar da testosterone a cikin marasa lafiya tare da ci-gaban ciwon daji na prostate lokacin da wasu zaɓuɓɓukan magani ke iyakance. Yana hana fitowar LH da FSH kai tsaye, wanda daga baya ya rage sakin testosterone daga ɗigon jini. Ta hanyar hana kwayoyin cutar kansar prostate na testosterone, abarelix yana taimakawa wajen kula da cutar da kuma kawar da alamun da ke hade.


Yin amfani da abarelix a cikin maganin ciwon gurguwar prostate yana ba da madaidaicin madadin ga marasa lafiya waɗanda ba za su iya sha ko ƙin simintin tiyata ko wasu magungunan hormonal ba. Ƙarfinsa na adawa da GnRH da kuma kawar da samar da testosterone yana ba da taimako na jin dadi kuma yana taimakawa wajen sarrafa ci gaban cutar. Ta hanyar rage matakan testosterone, abarelix yana taimakawa wajen hana ci gaba da yaduwar ƙwayoyin cutar kansar prostate, don haka yana ba da taimako na alamun bayyanar cututtuka da inganta yanayin rayuwar mai haƙuri.

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Abarelix, antagonist na hormone mai sakin gonadotropin, zaɓi ne mai mahimmanci na warkewa ga marasa lafiya da ke fama da ciwon daji na prostate wanda ba su dace da ƴan takara don luteinizing hormone-reaseing hormone agonists ko aikin tiyata ba. Ta hanyar hanawa LH da FSH kai tsaye, abarelix yana rage yawan samar da testosterone, wanda ke da mahimmanci ga ci gaba da ci gaban ciwon daji na prostate. Amfani da shi yana ba da taimako na jin daɗi kuma yana taimakawa sarrafa cutar a cikin marasa lafiya da ke da iyakataccen zaɓin magani. Abarelix, wanda aka sayar da shi azaman Plenaxis, yana aiki azaman kayan aiki mai mahimmanci a cikin yaƙi da ciwon daji na prostate mai ci gaba, yana ba da gudummawa ga ingantattun sakamakon haƙuri da ingantaccen rayuwa.
Ka tuna don tuntuɓar mu idan kuna da bukata.

Ƙayyadaddun bayanai

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