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Flumazenil A Zaɓaɓɓen Maganin Mai karɓar GABAA da Aikace-aikacen warkewa

Farashin Magana: USD 1-2/g

  • Sunan samfur Flumazenil
  • CAS No. 78755-81-4
  • MF Saukewa: C15H14FN3O3
  • MW 303.288363
  • EINECS 616-650-9
  • Yawan yawa 1.39
  • Wurin narkewa 201-203 ℃

Cikakken Bayani

Flumazenil, wanda kuma aka sani da flumazepil ko sunan lambar Ro 15-1788, zaɓin mai karɓar mai karɓar GABAA ne wanda za'a iya gudanar da shi ta hanyar allura, shigar da otic, ko ta cikin hanci. Yana aiki a matsayin duka antagonist da maganin maganin benzodiazepines, musamman a lokuta masu yawa, ta hanyar hanawa gasa. Wannan labarin yana bincika fa'idodin warkewa, amfani azaman maganin rigakafi, da yuwuwar aikace-aikacen flumazenil a cikin saitunan likita daban-daban.

I. Tsarin Aiki:
A. Zaɓaɓɓen GABAA antagonist
B. Hana gasa a wurin ganewar benzodiazepine
C. Juya tasirin benzodiazepine

II. Maganin rigakafin Benzodiazepine fiye da kima:
A. Muhimmancin hana gasa a cikin lokuta masu yawa
B. Fa'idodin flumazenil a cikin juyar da rashin jin daɗi da yawa
C. Matsaloli da haɗari masu alaƙa da amfani da kulawa mai tsanani
D. Abubuwan la'akari don yawan allurai da saka idanu a hankali

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III. Aikace-aikacen Bayan tiyata:

A. Komawar abubuwan kwantar da hankali na benzodiazepines bayan tiyata

B. Kwatankwacin amfani da naloxone a cikin juyawar opioid

C. Anesthesiologist saka idanu da la'akari bayan tiyata


IV. Jiyya na Ƙunƙasar Ƙunƙasar Ƙwararrun Ƙwararrun Ƙwararrun Ƙwararrun Ƙwararrun Ƙwararrun Ƙwararrun Ƙwararru:

A. Amfanin flumazenil wajen maganin zolpidem, zaleplon, da zopiclone overdoses


V. Aikace-aikace masu yuwuwa a cikin Hypersomnia da Tasirin Gastrointestinal:

A. Rage yawan barcin rana a hypersomnias na farko

B. Rage illolin da ke haifar da ciwon daji

C. Kariya na ƙwayoyin sel na hanji a lokacin chemotherapy da radiation far


VI. Muhimmancin Daidaita Hana Mai karɓar GABAA:

A. Kare ƙananan ƙwayoyin hanji daga lalacewar DNA yayin aikin rediyo

B. Tabbatar da kashe kwayoyin cutar daji ba a cikin damuwa



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Flumazenil, zaɓaɓɓen antagonist mai karɓa na GABAA, yana aiki azaman maganin rigakafi mai mahimmanci a cikin lokuta masu yawa na benzodiazepine, yana ba da gasa hanawa da jujjuya tasirin magani. Aikace-aikacen sa sun ƙara zuwa amfani da bayan tiyata, jiyya na marasa amfani da benzodiazepine hypnotic overdoses, da yuwuwar fa'idodi a cikin hypersomnia da sakamako masu illa na gastrointestinal. Kulawa a hankali da la'akari da haɗari suna da mahimmanci yayin gudanar da flumazenil, musamman a cikin tsananin kulawa da saitunan bayan tiyata. Ana buƙatar ƙarin bincike don gano cikakken ƙarfinsa don kare ƙwayoyin ƙwayoyin hanji yayin jiyya na ciwon daji tare da kiyaye tasirin cutar kansa.

Ƙayyadaddun bayanai

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