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Leuprorelin Hormone Therapy don Prostate da Cancer na Nono

Farashin: USD 30-100

  • Sunan samfur Leuprorelin
  • CAS No. 53714-56-0
  • Yawan yawa 1.44
  • Wurin narkewa 150-155 ° C
  • Wurin tafasa 1720.5°C a 760 mmHg
  • MF Saukewa: C59H84N16O12
  • MW 1269.473
  • Indexididdigar refractive 1.681
  • Ma'anar walƙiya 994.3°C

Cikakken Bayani

Leuprorelin, wanda kuma aka sani da Lupron ko Prostap, magani ne na hormone da ake amfani dashi don maganin prostate da ciwon nono. Yana cikin rukunin magunguna da ake kira gonadotropin-releasing hormone (GnRH) agonists. A cikin wannan maƙala, za mu mai da hankali kan amfani da ita wajen maganin cutar sankarar prostate da nono.

Maganin Ciwon Cutar Prostate:
Ana amfani da Leuprorelin don magance ciwon daji na prostate. Yana aiki ta hanyar rage matakin testosterone da ƙwai ke samarwa. Kwayoyin ciwon daji na prostate sun dogara da testosterone don girma, don haka rage matakansa zai iya rage ciwon daji ko rage girman girma. Gudanar da leuprorelin yana taimakawa wajen sarrafa alamun da ke hade da ciwon daji na prostate da kuma inganta yanayin rayuwar mai haƙuri.

Maganin Ciwon Kansa:
Hakanan ana amfani da Leuprorelin wajen maganin wasu nau'ikan ciwon daji na nono. An yi amfani da shi musamman a lokuta inda kwayoyin cutar kansa ke da masu karɓar isrogen (ER tabbatacce) kuma mai haƙuri bai shiga cikin menopause ba. Leuprorelin yana rage matakin estrogen a cikin jiki ta hanyar hana samar da shi a cikin ovaries. Wannan yana da mahimmanci saboda yawan isrogen na iya haɓaka haɓakar ƙwayoyin cutar kansar nono. Ana iya gudanar da Leuprorelin shi kaɗai ko a haɗe tare da wasu hanyoyin maganin hormone don sarrafa kansar nono yadda ya kamata.


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Balaga ta Tsakiyar Precocious:

Ana amfani da allurar Leuprorelin, wanda aka sani da Lupron Depot-PED, a cikin yara masu shekaru 2 da haihuwa don magance balaga ta tsakiya (CPP). CPP wani yanayi ne wanda 'yan mata (yawanci kasa da shekaru 8) da samari (yawanci kasa da shekaru 9) ke shiga balaga da wuri. Leuprorelin yana taimakawa wajen daidaita lokacin balaga ta hanyar rage saurin haɓakar ƙashi da haɓaka halayen jima'i da ke hade da CPP.


Sauran Amfanin Clinical:

Ana amfani da allurar Leuprorelin, wanda kuma aka sani da Lupron Depot, a cikin maganin endometriosis da anemia wanda fibroids na mahaifa ke haifarwa. Yana aiki ta hanyar rage matakan wasu hormones a cikin jiki, yana ba da taimako daga alamun cututtuka kamar zafi, nauyi ko rashin daidaituwa na haila, da anemia. Bugu da ƙari, ana iya amfani da leuprorelin a matsayin magani kafin magani na endometrial, kamar yadda ya rage ƙwayar endometrium, yana rage kumburi, kuma yana sauƙaƙe aikin tiyata.


Pharmacokinetics:
Leuprorelin acetate ba shi da tasiri idan an sha baki kuma a maimakon haka ana gudanar da shi ta hanyar allurar subcutaneous ko intramuscularly. Bayan allurar subcutaneous guda ɗaya na 3.75 MG, ana kaiwa ga mafi girman ƙwayar plasma a cikin kwanaki 1 zuwa 2, tare da matakan 1 zuwa 2 ng/ml. A cikin maganin ciwon daji na prostate, ana ba da allurar subcutaneous na 3.75 MG kowane mako 4 don jimlar allura 3 don cimma daidaiton matakan plasma na 0.1 zuwa 1 ng/ml. Leuprorelin yana metabolized zuwa samfuran lalacewa guda huɗu a cikin jiki kuma ana fitar dashi da farko ta cikin kodan.

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Ƙarshe:
Leuprorelin, GnRH agonist, magani ne mai mahimmanci na hormone wanda ake amfani dashi a maganin prostate da ciwon nono, da kuma tsakiyar precocious balaga, endometriosis, da anemia lalacewa ta hanyar fibroids uterine. Ta hanyar rage matakan testosterone ko estrogen, leuprorelin yana taimakawa wajen sarrafa girma da bayyanar cututtuka da ke hade da waɗannan yanayi. Gudanar da leuprorelin yana buƙatar kulawar likita da kulawa akai-akai don tabbatar da ingancinsa da sarrafa duk wani tasiri mai tasiri.

Ka tuna don tuntuɓar mu don cikakkun marufi da nau'ikan jigilar kaya, za mu samar da sabis na ƙwararrun OEM/ODM.

Ƙayyadaddun bayanai

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