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Telmisartan Mafi kyawun maganin hauhawar jini Kariyar koda

Farashin magana: USD 0.2-0.8/g

  • Sunan samfur Telmisartan
  • CAS No. 144701-48-4
  • MF Saukewa: C33H30N4O2
  • MW 514.629
  • EINECS 1592732-453-0

Cikakken Bayani

Telmisartan, wanda kuma aka sani da Timosartan, sabon magani ne mai rage hawan jini wanda aka keɓe azaman takamaiman mai karɓar mai karɓar angiotensin II (nau'in AT1). Ana amfani dashi sosai a cikin maganin hauhawar jini mai mahimmanci, yana ba da fa'idodi da yawa akan sauran magungunan antihypertensive. Wannan makalar tana da nufin samar da cikakken bayani game da fa'idodin Telmisartan da mahimman la'akari don amfani da shi.

Amfanin Telmisartan:

Mafi kyawun tasirin antihypertensive:
Telmisartan magani ne na farko na maganin hauhawar jini wanda aka saba wa wajabta saboda ingancinsa. A matsayin mai adawa da nau'in AT1, yana hana aikin angiotensin, yana haifar da raguwa mai yawa a cikin karfin jini. Telmisartan yana nuna matsayi mafi girma na musamman idan aka kwatanta da sauran sartans, yana ba shi damar shiga cikin membranes tantanin halitta da kuma ƙaddamar da takamaiman sel. Wannan ƙayyadaddun yana haɓaka tasirin sa na antihypertensive, yana haifar da raguwar hauhawar jini sosai. Bugu da ƙari, Telmisartan yana da tsawon rabin rayuwa, yana tabbatar da dorewa da ingantaccen sarrafa hawan jini.

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Kariyar tasoshin zuciya da jijiyoyin jini:

Telmisartan ya fito a matsayin kawai maganin sartan-kamar da FDA ta amince da shi don kariyar cututtukan zuciya da jijiyoyin jini. Yana nuna ikon juyar da hawan jini na hagu na hagu kuma ana ba da shawarar ga marasa lafiya da hauhawar jini tare da hauhawar jini na hagu, rashin isasshen zuciya, ko cututtukan jijiyoyin jini. Baya ga tasirinsa na rage hawan jini, Telmisartan yana rage lalacewar zuciya da jijiyoyin jini. Yana da amfani musamman ga mutanen da suka sami bugun jini ko ciwon zuciya.

Kare aikin koda:

Wani fa'idar Telmisartan shine tasirin sa mai kyau akan aikin koda. Tun da Telmisartan yana jure wa hanta metabolism kuma ana fitar dashi a cikin bile, yana da ƙarancin tasiri akan aikin koda. Hakanan, an gano Telmisartan don rage proteinuria, don haka yana kiyaye aikin koda. Yana da amfani musamman a cikin marasa lafiya masu fama da hauhawar jini da yanayin haɗuwa kamar su nephropathy na ciwon sukari, microalbuminuria, proteinuria, ko ƙarancin ƙarancin ƙima zuwa matsakaici.

Inganta juriya na insulin:

Telmisartan ya nuna ingantaccen tasiri akan metabolism na glucose da juriya na insulin. Wannan yanayin ya sa ya zama zaɓi mai dacewa ga marasa lafiya masu fama da hauhawar jini da ciwon sukari mellitus, saboda yana iya taimakawa haɓaka haɓakar insulin da sarrafa glucose.


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Telmisartan, takamaiman mai karɓar mai karɓar angiotensin II (nau'in AT1), yana ba da fa'idodi da yawa a cikin maganin hauhawar jini mai mahimmanci. Mafi kyawun sakamako na antihypertensive, kariya daga cututtukan zuciya da jijiyoyin jini, adana ayyukan koda, da haɓaka juriya na insulin ya sa ya zama zaɓi mai mahimmanci a cikin sarrafa hauhawar jini da yanayin alaƙa. Koyaya, yana da mahimmanci a bi ƙa'idodin shawarwari game da lokacin magani, sarrafa sashi, da saka idanu akai-akai don tabbatar da ingantaccen inganci da aminci. Ana ba da shawara tare da ƙwararrun kiwon lafiya koyaushe don shawarwari na keɓaɓɓu da jagora game da amfani da Telmisartan ko kowane magani.

Ƙayyadaddun bayanai

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