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ʻO Abarelix Power Gonadotropin-Hoʻokuʻu Hormone Antagonist no ka mālama ʻana i ka maʻi maʻi prostate

Kumukuai kuhikuhi: USD 100-200/g

  • inoa mea kūʻai Abarelix
  • CAS No. 183552-38-7
  • MF C72H95ClN14O14
  • MW 1416.0631
  • EINECS 1592732-453-0
  • ʻO ka mānoanoa 1.286
  • Lae paila 1688.4°Cat760mmHg
  • Kuhikuhi uila 974.9°C

Ka wehewehe kikoʻī

ʻO Abarelix, kahi decapeptide synthetic, hōʻike i ka hana antagonistic ikaika e kūʻē i ka hormone hoʻokuʻu gonadotropin-releasing hormone (GnRH). Hoʻohana mua ʻia ia e mālama i nā maʻi me ka maʻi prostate hōʻailona holomua ʻaʻole kūpono i nā moho no ka luteinizing hormone-releasing hormone agonists a i ʻole castration surgical. Ma ke kāohi pololei ʻana i ka huna ʻana o ka hormone luteinizing (LH) a me ka follicle-stimulating hormone (FSH), hoʻemi maikaʻi ʻo abarelix i ka hana ʻana o ka testosterone mai nā testicles. e ʻimi i nā hōʻailona therapeutic, nā ʻano hana, a me ka hoʻohana ʻana i ka abarelix.

Hōʻike ʻia ʻo Abarelix no ka mālama palliative o nā maʻi maʻi maʻi me ka maʻi maʻi prostate kiʻekiʻe e kū ana i nā koina kikoʻī. Manaʻo ʻia no nā poʻe maʻi ʻaʻole kūpono i nā moho no ka luteinizing hormone-releasing hormone agonists, hōʻole i ka castration surgical, a loaʻa i nā mea pilikia ʻē aʻe e like me ka hiki ke hōʻeha i ka neurological ma muli o ka metastasis, ureteral a i ʻole ʻākea orifice obstruction ma muli o ka erosion kūloko a i ʻole metastasis, a i ʻole ʻeha iwi metastatic koʻikoʻi e koi ana i ka hoʻomaha ʻana i ka ʻeha narcotic.


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Ma ke ʻano he gonadotropin-releasing hormone antagonist (GnRH antagonist), he hana koʻikoʻi ka abarelix i ka hōʻemi ʻana i ka hana ʻana o ka testosterone i nā poʻe maʻi me ka maʻi maʻi prostate maʻi maʻi ke kaupalena ʻia nā koho lapaʻau ʻē aʻe. Hoʻopili pololei ia i ka huna ʻana o LH a me FSH, a laila hoʻemi i ka hoʻokuʻu ʻana o ka testosterone mai nā testicles. Ma ka hoʻonele ʻana i nā maʻi maʻi prostate o ka testosterone, kōkua ʻo abarelix i ka mālama ʻana i ka maʻi a me ka hoʻohaʻahaʻa ʻana i nā hōʻailona pili.


ʻO ka hoʻohana ʻana i ka abarelix i ka mālama ʻana i ka maʻi maʻi prostate e hāʻawi i kahi koho koʻikoʻi no nā poʻe maʻi ʻaʻole hiki ke hoʻopaʻa a hōʻole paha i ka castration ʻoki a i ʻole nā ​​​​hopena hormonal. ʻO kona hiki ke kū'ē i ka GnRH a hoʻopaʻa i ka hana testosterone hāʻawi i ka hōʻoluʻolu palliative a kōkua i ka mālama ʻana i ka holomua o ka maʻi. Ma ka hōʻemi ʻana i nā pae testosterone, kōkua ka abarelix i ke kāohi ʻana i ka ulu a me ka hoʻonui ʻana o nā maʻi maʻi prostate, no laila e hāʻawi ana i ka hōʻoluʻolu hōʻailona a hoʻomaikaʻi i ka maikaʻi o ke ola o ka mea maʻi.

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ʻO Abarelix, he mea hoʻokuʻu ʻana i ka hormone antagonist ikaika, he koho therapeutic waiwai no nā poʻe maʻi me ka maʻi maʻi prostate hōʻailona holomua ʻaʻole kūpono i nā moho no ka luteinizing hormone-releasing hormone agonists a i ʻole castration surgical. Ma ka pale pololei ʻana i ka huna ʻana o LH a me FSH, hoʻemi maikaʻi ʻo abarelix i ka hana testosterone, he mea nui ia no ka ulu a me ka holomua o ka maʻi prostate. Hāʻawi kona hoʻohana ʻana i ka hōʻoluʻolu palliative a kōkua i ka mālama ʻana i ka maʻi i nā maʻi me nā koho lapaʻau liʻiliʻi. ʻO Abarelix, i kūʻai ʻia e like me Plenaxis, he mea hana koʻikoʻi i ka hakakā ʻana i ka maʻi maʻi prostate holomua, e hāʻawi ana i ka hoʻomaikaʻi ʻana i nā hopena maʻi a me ka maikaʻi o ke ola.
E hoʻomanaʻo e launa pū me mākou inā pono.

Hōʻike

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