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ʻO Telmisartan ʻoi aku ka maikaʻi o ka antihypertensive pale i ka renal

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  • inoa mea kūʻai Telmisartan
  • CAS No. 144701-48-4
  • MF C33H30N4O2
  • MW 514.629
  • EINECS 1592732-453-0

Ka wehewehe kikoʻī

ʻO Telmisartan, ka mea i kapa ʻia ʻo Timosartan, he lāʻau hoʻohaʻahaʻa koko koko hou i helu ʻia ma ke ʻano he angiotensin II receptor (AT1-type) antagonist. Hoʻohana nui ʻia ia i ka mālama ʻana i ka hypertension koʻikoʻi, e hāʻawi ana i nā pono he nui ma mua o nā lāʻau antihypertensive ʻē aʻe. Ke manaʻo nei kēia ʻatikala e hāʻawi i kahi ʻike piha o nā pono o Telmisartan a me nā noʻonoʻo koʻikoʻi no kāna hoʻohana.

ʻO nā mea maikaʻi o Telmisartan:

ʻOi aku ka hopena antihypertensive:
ʻO Telmisartan kahi lāʻau antihypertensive laina mua i kuhikuhi ʻia ma muli o kona kiʻekiʻe kiʻekiʻe. Ma ke ʻano he ʻano antagonist AT1, ke kāohi nei ia i ka hana o ka angiotensin, ka hopena i kahi hōʻemi nui o ke koko. Hōʻike ʻo Telmisartan i kahi kiʻekiʻe kiʻekiʻe o ka kikoʻī i hoʻohālikelike ʻia me nā sartans ʻē aʻe, e ʻae iā ia e komo maʻalahi i nā membrane cell a kuhikuhi i nā cell kikoʻī. Hoʻonui kēia kikoʻī i kāna mau hopena antihypertensive, e alakaʻi ana i kahi emi nui o ke koko. Eia kekahi, ʻoi aku ka lōʻihi o ka hapalua o ke ola ʻo Telmisartan, e hōʻoiaʻiʻo ana i ka hoʻomau ʻana a me ka maikaʻi o ke kahe koko.

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Ka pale ʻana i nā moku cardiovascular a me ka cerebral:

Kūʻē ʻo Telmisartan ʻo ia wale nō ka lāʻau e like me ka sartan i ʻae ʻia e ka FDA no kāna mau mea pale cardiovascular a me ka cerebrovascular. Hōʻike ia i ka hiki ke hoʻohuli i ka hypertrophy ventricular hema a ua ʻōlelo ʻia no nā poʻe maʻi me ka hypertension i hele pū ʻia me ka hypertrophy ventricular hema, ka lawa ʻole o ka naʻau, a i ʻole ka maʻi ʻaʻa coronary. Ma kahi o kāna mau hopena hoʻohaʻahaʻa i ke koko, hōʻemi ʻo Telmisartan i ka pōʻino cardiovascular a me cerebrovascular. He mea maikaʻi loa ia no ka poʻe i loaʻa i ka maʻi ʻaʻai a i ʻole ka maʻi puʻuwai.

Ka pale ʻana i ka hana renal:

ʻO kekahi pono ʻē aʻe o Telmisartan ʻo kona hopena maikaʻi i ka hana renal. No ka mea e hele ana ʻo Telmisartan i ka metabolism hepatic a hoʻokuʻu ʻia i loko o ka bile, he liʻiliʻi ka hopena i ka hana renal. Eia kekahi, ua ʻike ʻia ʻo Telmisartan e hōʻemi i ka proteinuria, ma laila e pale ai i ka hana renal. He mea pono loa ia i nā poʻe maʻi me ke kiʻekiʻe kiʻekiʻe a me nā kūlana comorbid e like me ka nephropathy diabetic, microalbuminuria, proteinuria, a i ʻole ka liʻiliʻi a i ʻole ka lawa ʻole o ka renal.

Ka hoʻomaikaʻi ʻana i ka pale ʻana i ka insulin:

Ua hōʻike ʻo Telmisartan i nā hopena maikaʻi i ka metabolism glucose a me ka pale ʻana i ka insulin. ʻO kēia hiʻohiʻona he koho kūpono ia no nā poʻe maʻi me ka hypertension a me ka maʻi diabetes mellitus, no ka mea hiki ke kōkua i ka hoʻomaikaʻi ʻana i ka ʻike insulin a me ka hoʻokele glucose.


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ʻO Telmisartan, kahi antagonist angiotensin II kikoʻī (AT1-type) antagonist, hāʻawi i nā pono he nui i ka mālama ʻana i ka hypertension koʻikoʻi. ʻO kāna hopena antihypertensive ʻoi aku ka maikaʻi, ka pale ʻana i nā kīʻaha cardiovascular a me ka cerebral, mālama i ka hana renal, a me ka hoʻomaikaʻi ʻana i ka insulin resistance e lilo ia i koho koʻikoʻi i ka mālama ʻana i ka hypertension a me nā kūlana pili. Eia nō naʻe, he mea koʻikoʻi ia e hahai i nā alakaʻi i ʻōlelo ʻia e pili ana i ka manawa o ka lāʻau lapaʻau, ka mālama ʻana i ka dosage, a me ka nānā mau ʻana e hōʻoia i ka maikaʻi a me ka palekana. Hoʻomaopopo mau ʻia ke kūkākūkā me kahi ʻoihana mālama ola no ka ʻōlelo aʻoaʻo pilikino a me ke alakaʻi e pili ana i ka hoʻohana ʻana iā Telmisartan a i ʻole kekahi lāʻau lapaʻau.

Hōʻike

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