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Telmisartan Zoo dua antihypertensive Tiv thaiv lub raum

Nqe: USD 0.2-0.8 / g

  • Khoom npe Telmisartan
  • CAS Nr. 144701-48-4
  • MF C33H30N4O2
  • MW 514.629 ib
  • EINECS 1592732-453-0

Cov lus piav qhia ntxaws

Telmisartan, tseem hu ua Timosartan, yog cov tshuaj tshiab ntshav siab-txo cov tshuaj cais raws li cov tshuaj angiotensin II receptor (AT1-type) antagonist. Nws yog dav siv nyob rau hauv kev kho mob ntawm qhov tseem ceeb kub siab, muab ntau yam zoo dua lwm cov tshuaj antihypertensive. Tsab ntawv no yog npaj los muab cov lus qhia dav dav ntawm cov txiaj ntsig ntawm Telmisartan thiab cov kev xav tseem ceeb rau nws siv.

Qhov zoo ntawm Telmisartan:

Cov nyhuv antihypertensive zoo dua:
Telmisartan yog ib hom tshuaj tiv thaiv kab mob siab tshaj plaws hauv thawj kab vim nws cov txiaj ntsig zoo. Raws li AT1-hom antagonist, nws inhibits qhov kev txiav txim ntawm angiotensin, ua rau txo qis ntshav siab. Telmisartan nthuav tawm ntau dua ntawm qhov tshwj xeeb piv rau lwm cov sartans, tso cai rau nws yooj yim nkag mus rau cov cell membranes thiab lub hom phiaj tshwj xeeb. Qhov tshwj xeeb no txhim kho nws cov teebmeem antihypertensive, ua rau txo qis ntshav siab ntau. Tsis tas li ntawd, Telmisartan muaj ib nrab-lub neej ntev, ua kom cov ntshav siab tswj tau zoo.

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Kev tiv thaiv kab mob plawv thiab hlab ntsha hlwb:

Telmisartan sawv tawm raws li cov tshuaj sartan nkaus xwb pom zoo los ntawm FDA rau nws cov hlab plawv thiab cerebrovascular tiv thaiv. Nws qhia tau hais tias muaj peev xwm thim rov qab sab laug ventricular hypertrophy thiab pom zoo rau cov neeg mob ntshav siab nrog rau sab laug ventricular hypertrophy, plawv tsis txaus, lossis kab mob plawv. Ntxiv nrog rau nws cov ntshav siab-txo cov teebmeem, Telmisartan txo cov hlab plawv thiab cerebrovascular puas. Nws yog qhov tshwj xeeb tshaj yog rau cov tib neeg uas tau ntsib kev mob stroke lossis plawv infarction.

Tiv thaiv lub raum ua haujlwm:

Lwm qhov zoo dua ntawm Telmisartan yog nws cov txiaj ntsig zoo rau lub raum ua haujlwm. Txij li Telmisartan dhau los ua cov metabolism hauv hepatic thiab raug tso tawm hauv cov kua tsib, nws muaj kev cuam tshuam tsawg rau lub raum ua haujlwm. Ntxiv mus, Telmisartan tau pom tias txo cov proteinuria, yog li tiv thaiv lub raum ua haujlwm. Nws yog tshwj xeeb tshaj yog pab tau rau cov neeg mob ntshav siab thiab comorbid tej yam kev mob xws li mob ntshav qab zib nephropathy, microalbuminuria, proteinuria, los yog me me mus rau nruab nrab lub raum tsis txaus.

Kev txhim kho ntawm insulin tsis kam:

Telmisartan tau pom tias muaj txiaj ntsig zoo rau cov metabolism hauv qabzib thiab insulin tsis kam. Cov yam ntxwv no ua rau nws muaj kev xaiv tsim nyog rau cov neeg mob ntshav siab thiab ntshav qab zib mellitus, vim nws tuaj yeem pab txhim kho insulin rhiab heev thiab tswj cov piam thaj.


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Telmisartan, ib qho tshwj xeeb angiotensin II receptor (AT1-type) antagonist, muaj ntau yam zoo hauv kev kho mob ntshav siab tseem ceeb. Nws cov nyhuv antihypertensive zoo dua, kev tiv thaiv cov hlab plawv thiab cov hlab ntsha hauv hlwb, khaws cia lub raum ua haujlwm, thiab txhim kho cov tshuaj insulin ua rau nws muaj txiaj ntsig zoo rau kev tswj ntshav siab thiab cov xwm txheej cuam tshuam. Txawm li cas los xij, nws yog ib qho tseem ceeb uas yuav tsum ua raws li cov lus pom zoo hais txog lub sij hawm siv tshuaj, kev tswj kev noj tshuaj, thiab kev saib xyuas tsis tu ncua kom ntseeg tau tias kev ua tau zoo thiab kev nyab xeeb. Kev sab laj nrog tus kws kho mob yeej ib txwm qhia rau tus kheej cov lus qhia thiab kev taw qhia txog kev siv Telmisartan lossis txhua yam tshuaj.

Specification

17165252945776 jr