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Dapoxetine ntụ ntụ mbadamba Dapoxetine Premature Ejaculation na Men

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  • Aha ngwaahịa Dapoxetine
  • Ọdịdị Uzuzu crystalline na-acha ọcha ruo na-acha ọcha
  • CAS Mba. 119356-77-3
  • MF C21H23NO
  • MW 305.41300
  • Njupụta 1.081 g/cm3
  • Ebe esi nri 454.4ºC na 760mmHg
  • ebe mgbari 132.6ºC
  • Ntụgharị ntụgharị 1.607

Nkọwa zuru ezu

Dapoxetine, CAS No. 119356-77-3, na usoro molecular C21H23NO, bụ ọgwụ eji eme ihe maka ọgwụgwọ ejaculation akaghi aka na ụmụ nwoke. Ọ na-apụta dị ka ntụ ntụ crystalline na-acha ọcha ma na-acha ọcha, ọ naghịkwa isi ísì. Dapoxetine nwere oke solubility na mmiri.

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Dapoxetine ntụ ntụ bụ ụdị ọhụrụ SSRI ngwa ngwa na obere ọkara ndụ. Ọ bụ onye na-emechi ihe nchịkwa nke serotonin (SSRI). Ọ bụ ọgwụ eji agwọ ejaculation akaghi aka n'ime ụmụ nwoke dị afọ 16 ruo 84.

N'ime usoro ọmụmụ ihe akaebe nke abụọ nke PPD mere, dapoxetine gosipụtara mmụba dị ịrịba ama na njedebe ejaculatory ma e jiri ya tụnyere placebo. otutu dosing.
Eserese ọrụ u3g


Dapoxetine (INN, akara aha Priligy), ụdị usoro ọgwụgwọ a na-ejikarị bụ mbadamba, anyị na-akwadokwa capsules ahaziri. N'ịbụ nke e mepụtara dị ka antidepressant, e mesịrị chọpụta na ọ nwekwara mmetụta dị mma n'ịgwọ ejaculation akaghi aka (PE). A na-ewere ya ugbu a dị ka ọgwụgwọ dị irè maka ejaculation akaghi aka na ụmụ nwoke. Dapoxetine nwere ike ịgbatị oge nke mmekọahụ na ụmụ nwoke, si otú a na-eme ka ndụ ha dịkwuo mma. Dapoxetine na-agbanwe ntụgharị akwara site na igbochi reuptake nke serotonin, si otú a na-amụba ntinye nke serotonin na synapses. Omume a na-enye ohere dapoxetine ịgbatị ogologo oge nke mmekọahụ, si otú a na-enyere ndị ikom na-ata ahụhụ site na nsogbu ejaculation akabeghị aka. Usoro ọgwụgwọ nke dapoxetine na-abụkarị 30mg ma ọ bụ 60mg, nke nwere ike gbanwee dịka ọnọdụ onye ọrịa siri dị. A na-etinye ya ngwa ngwa mgbe nchịkwa ọnụ gasịrị, ọ na-ewe ihe dịka awa 1-2 iji rute mkpokọta plasma kacha elu. Ọkara ndụ nke dapoxetine bụ ihe dị ka awa 1-2, nke pụtara na ọ na-emepụta ma na-apụ ngwa ngwa n'ime ahụ. N'ọtụtụ ndị ọrịa, iji dapoxetine dị mma, ma ụfọdụ mmeghachi omume ọjọọ nwere ike ime, gụnyere isi ọwụwa, ọgbụgbọ, ehighi ura, ike ọgwụgwụ, wdg. Tupu ịmalite dapoxetine, ị kwesịrị ịgwa dọkịta gị okwu iji jide n'aka na ọ dịghị ihe ize ndụ nke mmekọrịta gị na ndị ọzọ. ọgwụ ma ọ bụ ọnọdụ ahụike dị adị.

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