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Flumazenil A Nhọrọ GABAA Nnabata Onye Mmegide na Ngwa Ọgwụ Ya

Ọnụ ego ntụaka: USD 1-2/g

  • Aha ngwaahịa Flumazenil
  • CAS Mba. 78755-81-4
  • MF C15H14FN3O3
  • MW 303.288363
  • EINECS 616-650-9
  • Njupụta 1.39
  • Ebe mgbaze 201-203 ℃

Nkọwa zuru ezu

Flumazenil, nke a makwaara dị ka flumazepil ma ọ bụ koodu aha Ro 15-1788, bụ onye na-anabata GABAA antagonist nke enwere ike ịnye ya site na ntụtụ, ntinye otic, ma ọ bụ intranasally. Ọ na-eme dị ka ma onye na-emegide ya na ọgwụ mgbochi benzodiazepines, karịsịa n'ihe banyere ịṅụbiga mmanya ókè, site na mgbochi asọmpi. Edemede a na-enyocha uru ọgwụgwọ, ojiji dị ka ọgwụ mgbochi, yana ngwa nwere ike iji flumazenil na ntọala ahụike dị iche iche.

I. Usoro nke Omume:
A. Nhọrọ GABAA antagonist
B. Mgbochi asọmpi na saịtị njirimara benzodiazepine
C. Mweghachi mmetụta benzodiazepine

II. Ngwọta maka Benzodiazepine Ngafe:
A. Mkpa nke mgbochi asọmpi n'ihe gbasara ịṅụbiga mmanya ókè
B. Uru nke flumazenil n'ịgbanwe oke ịhịa aka n'ahụ
C. Mgbagwoju anya na ihe egwu jikọtara ya na nnukwu nlekọta nlekọta
D. Atụmatụ maka otutu dosing na nlezianya nlekota

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III. Ngwa gbasara ịwa ahụ:

A. Mgbanwe nke mmetụta ịhịa aka n'ahụ nke benzodiazepines mgbe a wachara ya ahụ

B. Myirịta na ojiji naloxone na ngbanwe opioid

C. Anesthesiologist nlekota na echiche post-ịwa ahụ


IV. Ọgwụgwọ nke na-abụghị Benzodiazepine Hypnotic overdoses:

A. Ịdị irè nke flumazenil na ọgwụgwọ zolpidem, zaleplon, na zopiclone.


V. Ngwa nwere ike na Hypersomnia na Mmetụta Akụkụ Gastrointestinal:

A. Mbelata oke ụra nke ụbọchị na hypersomnias nke mbụ

B. Mbelata mmetụta nke eriri afọ nke ọgwụgwọ ọrịa kansa kpatara

C. Nchekwa mkpụrụ ndụ eriri afọ n'oge chemotherapy na ọgwụgwọ radieshon


VI. Mkpa nke imezi ihe mgbochi GABAA nnabata:

A. Chebe mkpụrụ ndụ eriri afọ site na mmebi DNA n'oge ọgwụgwọ redio

B. Ịhụ na igbu mkpụrụ ndụ kansa adịghị emebi emebi



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Flumazenil, onye na-anabata onye na-anabata GABAA, na-eje ozi dị ka ọgwụ bara uru na benzodiazepine ịdoụbiga mmanya ókè, na-enye mgbochi asọmpi na ngbanwe nke mmetụta ọgwụgwọ. Ngwa ya na-agbatị ruo mgbe ịwa ahụ gasịrị, ọgwụgwọ nke na-abụghị benzodiazepine hypnotic overdoses, na uru nwere ike na hypersomnia na eriri afọ mmetụta. Nleba anya nke ọma na nleba anya nke ihe egwu dị mkpa mgbe ị na-enye flumazenil, ọkachasị na nlekọta ahụike na ntọala ịwa ahụ. Achọrọ nyocha ọzọ iji chọpụta ikike ya zuru oke n'ichekwa mkpụrụ ndụ eriri afọ n'oge ọgwụgwọ ọrịa kansa ka ọ na-ejigide nrụpụta mkpụrụ ndụ kansa na-egbu egbu.

Nkọwapụta

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