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Flumazenil A Selective GABAA Receptor Antagonist ndi Therapeutic Applications

Mtengo Wolozera:USD 1-2/g

  • Dzina lazogulitsa Flumazenil
  • CAS No. 78755-81-4
  • MF Chithunzi cha C15H14FN3O3
  • MW 303.288363
  • Malingaliro a kampani EINECS 616-650-9
  • Kuchulukana 1.39
  • Malo osungunuka 201-203 ℃

Kufotokozera Mwatsatanetsatane

Flumazenil, yemwe amadziwikanso kuti flumazepil kapena code name Ro 15-1788, ndi wosankha GABAA receptor antagonist yemwe amatha kuperekedwa kudzera mu jakisoni, kuyika otic, kapena intranasally. Imakhala ngati wotsutsa komanso antidote kwa benzodiazepines, makamaka pazochitika za overdose, chifukwa cha mpikisano woletsa. Nkhaniyi ikufotokoza za ubwino wachirengedwe, kugwiritsidwa ntchito ngati mankhwala, komanso kugwiritsa ntchito kwa flumazenil m'malo osiyanasiyana azachipatala.

I. Kachitidwe Kachitidwe:
A. Selective GABAA receptor antagonist
B. Kuletsa mpikisano pamalo ozindikira benzodiazepine
C. Kusintha kwa zotsatira za benzodiazepine

II. Antidote kwa Benzodiazepine Overdose:
A. Kufunika koletsa mpikisano pamilandu ya bongo
B. Ubwino wa flumazenil pochepetsa kukomoka kwambiri
C. Zovuta ndi zoopsa zomwe zimagwirizanitsidwa ndi kugwiritsidwa ntchito kwachisamaliro
D. Kuganizira za madontho angapo ndi kuwunika mosamala

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III. Kugwiritsa Ntchito Pambuyo pa Opaleshoni:

A. Kusintha kwa sedative zotsatira za benzodiazepines pambuyo pa opaleshoni

B. Zofanana ndi kugwiritsa ntchito kwa naloxone mukusintha kwa opioid

C. Kuwunika kwa Anesthesiologist ndi kuganizira pambuyo pa opaleshoni


IV. Chithandizo cha Non-Benzodiazepine Hypnotic Overdoses:

A. Kuchita bwino kwa flumazenil pochiza zolpidem, zaleplon, ndi zopiclone overdose


V. Ntchito Zomwe Zingachitike mu Hypersomnia ndi Zotsatira Zam'mimba:

A. Kuchepetsa kugona mopitirira muyeso masana mu primary hypersomnias

B. Kuchepetsa zotsatira za m'mimba chifukwa cha mankhwala a khansa

C. Chitetezo cha m'matumbo tsinde maselo pa chemotherapy ndi ma radiation therapy


VI. Kufunika kwa Kulinganiza GABAA Receptor Inhibition:

A. Kuteteza maselo a m'matumbo ku kuwonongeka kwa DNA panthawi ya radiotherapy

B. Kuwonetsetsa kuti kupha maselo a khansa sikusokonezedwa



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Flumazenil, wosankha GABAA receptor antagonist, amagwira ntchito ngati mankhwala othandiza kwambiri pamilandu ya benzodiazepine overdose, kupereka kuletsa kwapikisano komanso kubweza zotsatira za sedative. Kugwiritsa ntchito kwake kumafikira kugwiritsidwa ntchito pambuyo pa opaleshoni, chithandizo chamankhwala osagwiritsa ntchito benzodiazepine hypnotic overdose, komanso mapindu omwe angakhalepo mu hypersomnia ndi zotsatira za m'mimba. Kuyang'anira mosamala ndikuwunika zoopsa ndikofunikira popereka flumazenil, makamaka pakasamalidwe koopsa komanso pambuyo pa opaleshoni. Kafukufuku wowonjezereka akufunika kuti afufuze momwe angathere poteteza maselo am'mimba panthawi ya chithandizo cha khansa ndikusunga mphamvu yakupha maselo a khansa.

Kufotokozera

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