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Telmisartan Bwino antihypertensive Kuteteza aimpso

Mtengo wolozera: USD 0.2-0.8/g

  • Dzina lazogulitsa Telmisartan
  • CAS No. 144701-48-4
  • MF Chithunzi cha C33H30N4O2
  • MW 514.629
  • Malingaliro a kampani EINECS 1592732-453-0

Kufotokozera Mwatsatanetsatane

Telmisartan, yomwe imadziwikanso kuti Timosartan, ndi mankhwala atsopano ochepetsa kuthamanga kwa magazi omwe amadziwika kuti ndi mdani wina wa angiotensin II receptor (mtundu wa AT1). Amagwiritsidwa ntchito kwambiri pochiza matenda oopsa kwambiri, omwe amapereka zabwino zingapo kuposa mankhwala ena a antihypertensive. Nkhaniyi ikufuna kupereka chiwongolero chonse chazabwino za Telmisartan ndi zofunikira pakugwiritsa ntchito kwake.

Ubwino wa Telmisartan:

Ubwino wa antihypertensive effect: +
Telmisartan ndi mankhwala omwe nthawi zambiri amaperekedwa pamzere woyamba wa antihypertensive chifukwa champhamvu kwambiri. Monga wotsutsa wamtundu wa AT1, amalepheretsa zochita za angiotensin, zomwe zimapangitsa kuchepa kwakukulu kwa kuthamanga kwa magazi. Telmisartan imawonetsa mulingo wapamwamba kwambiri poyerekeza ndi ma sartan ena, kuwalola kuti azitha kulowa mu nembanemba yama cell ndikulunjika ma cell enieni. Izi zimakulitsa zotsatira zake za antihypertensive, zomwe zimapangitsa kuti kuthamanga kwa magazi kuchepe. Kuphatikiza apo, Telmisartan imakhala ndi theka la moyo wautali, kuwonetsetsa kuti kuthamanga kwa magazi kumakhazikika komanso kogwira mtima.

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Kuteteza ziwiya zamtima ndi ubongo:

Telmisartan imadziwika kuti ndi mankhwala okhawo okhala ngati sartan omwe amavomerezedwa ndi FDA chifukwa chachitetezo chake chamtima komanso cerebrovascular. Imawonetsa kuthekera kosinthira kumanzere kwamitsempha yamagazi hypertrophy ndipo imalimbikitsidwa kwa odwala omwe ali ndi matenda oopsa omwe amatsagana ndi kumanzere kwa ventricular hypertrophy, kulephera kwamtima, kapena matenda a mtima. Kuphatikiza pa kutsika kwake kwa kuthamanga kwa magazi, Telmisartan imachepetsa kuwonongeka kwamtima ndi cerebrovascular. Ndiwothandiza makamaka kwa anthu omwe adakumana ndi stroke kapena mtima infarction.

Kuteteza aimpso ntchito:

Ubwino wina wa Telmisartan ndikuti imakhudzanso ntchito yaimpso. Popeza Telmisartan imalowa m'chiwindi ndipo imatulutsidwa mu bile, imakhudza kwambiri aimpso. Kuphatikiza apo, Telmisartan yapezeka kuti imachepetsa proteinuria, motero imateteza aimpso kugwira ntchito. Ndiwothandiza makamaka kwa odwala matenda oopsa komanso comorbid mikhalidwe monga diabetesic nephropathy, microalbuminuria, proteinuria, kapena kulephera kwaimpso pang'ono kapena pang'ono.

Kuchulukitsa kwa insulin kukana: +

Telmisartan yawonetsa zotsatira zabwino pa metabolism ya glucose komanso kukana insulini. Khalidweli limapangitsa kukhala njira yoyenera kwa odwala omwe ali ndi matenda oopsa komanso matenda a shuga, chifukwa amathandizira kukulitsa chidwi cha insulin komanso kuwongolera shuga.


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Telmisartan, wotsutsa wa angiotensin II receptor (mtundu wa AT1) amapereka zabwino zingapo pochiza matenda oopsa kwambiri. Mphamvu yake yabwino ya antihypertensive, kuteteza mtima ndi mitsempha yamagazi, kuteteza aimpso, komanso kusintha kwa insulin kukana kumapangitsa kukhala chisankho chofunikira pakuwongolera kuthamanga kwa magazi ndi zovuta zina. Komabe, ndikofunikira kutsatira malangizo okhudzana ndi nthawi yamankhwala, kuwongolera mlingo, komanso kuwunika pafupipafupi kuti muwonetsetse kuti ali ndi mphamvu komanso chitetezo chokwanira. Kukaonana ndi dokotala kumalangizidwa nthawi zonse kuti mupeze upangiri wamunthu payekha komanso chitsogozo chokhudza kugwiritsa ntchito Telmisartan kapena mankhwala aliwonse.

Kufotokozera

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