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Flumazenil Yatoranijwe GABAA yakira Antagonist hamwe nuburyo bwo kuvura

Igiciro Reba: USD 1-2 / g

  • izina RY'IGICURUZWA Flumazenil
  • URUBANZA No. 78755-81-4
  • MF C15H14FN3O3
  • MW 303.288363
  • EINECS 616-650-9
  • Ubucucike 1.39
  • Ingingo yo gushonga 201-203 ℃

Ibisobanuro birambuye

Flumazenil, izwi kandi nka flzwepil cyangwa izina rya kode Ro 15-1788, ni antagonist ya GABAA yatoranijwe ishobora gutangwa hakoreshejwe inshinge, kwinjiza otic, cyangwa imbere. Ikora nka antagonist na antidote kuri benzodiazepine, cyane cyane mugihe kirenze urugero, binyuze mukubuza guhatana. Iyi ngingo iragaragaza inyungu zo kuvura, ikoreshwa nka antidote, hamwe nibishobora gukoreshwa na flumazenil mubuvuzi butandukanye.

I. Uburyo bwibikorwa:
A. Guhitamo GABAA yakira antagonist
B. Kubuza guhiganwa kurubuga rwa benzodiazepine
C. Guhindura ingaruka za benzodiazepine

II. Umuti urwanya Benzodiazepine Kurenza urugero:
A. Akamaro ko kubuza guhatanira kurenza urugero
B. Inyungu za flumazenil muguhindura imitekerereze ikabije
C. Ingorane n'ingaruka zijyanye no gukoresha ubuvuzi bukabije
D. Ibitekerezo byo gufata inshuro nyinshi no gukurikirana neza

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III. Gusaba nyuma yo kubagwa:

A. Guhindura ingaruka ziterwa na benzodiazepine nyuma yo kubagwa

B. Ibisa no gukoresha naloxone muguhindura opioid

C. Gukurikirana Anesthesiologue no gutekereza nyuma yo kubagwa


IV. Umuti wa Hypnotic Hypnotic Non-Benzodiazepine:

A. Ingaruka za flumazenil mukuvura zolpidem, zaleplon, na zopiclone birenze urugero


V. Ibishobora gukoreshwa muri Hypersomnia na Gastrointestinal Side Ingaruka:

A. Kugabanya ibitotsi byinshi kumanywa muri hypersomnias yibanze

B. Kugabanya ingaruka mbi za gastrointestinal ziterwa no kuvura kanseri

C. Kurinda ingirangingo zo munda mugihe cya chimiotherapie no kuvura imirasire


VI. Akamaro ko Kuringaniza GABAA Kwakira Kwakira:

A. Kurinda ingirangingo zo munda kwangirika kwa ADN mugihe cya radiotherapi

B. Kureba ko kwica kanseri ya kanseri bitabangamiwe



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Flumazenil, antagonist ya GABAA yatoranijwe, ikora nk'umuti urwanya indwara ya benzodiazepine ikabije, itanga uburyo bwo kubuza irushanwa no guhindura ingaruka ziterwa no kwikuramo. Porogaramu zayo zikoreshwa nyuma yo kubagwa, kuvura hypnotic hypnotic itari benzodiazepine, hamwe ninyungu zishobora guterwa na hypersomnia n'ingaruka za gastrointestinal. Gukurikirana neza no gusuzuma ingaruka ni ngombwa mugihe utanga flumazenil, cyane cyane mubuvuzi bukabije ndetse na nyuma yo kubagwa. Ubushakashatsi burakenewe kugira ngo hamenyekane imbaraga zabwo zose mu kurinda ingirangingo zo mu nda mu gihe cyo kuvura kanseri mu gihe hakomeza kubaho ingaruka zo kwica kanseri.

Ibisobanuro

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