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Leuprorelin Hormone ivura Kanseri ya Prostate na Amabere

Igiciro cyerekana: USD 30-100

  • Izina RY'IGICURUZWA Leuprorelin
  • URUBANZA No. 53714-56-0
  • Ubucucike 1.44
  • Ingingo yo gushonga 150-155 ° C.
  • Ingingo yo guteka 1720.5 ° C kuri 760 mmHg
  • MF C59H84N16O12
  • MW 1269.473
  • Ironderero 1.681
  • Ingingo ya Flash 994.3 ° C.

Ibisobanuro birambuye

Leuprorelin, izwi kandi nka Lupron cyangwa Prostap, ni imiti ivura imisemburo ikoreshwa mu kuvura kanseri ya prostate na kanseri y'ibere. Ni mubyiciro byimiti yitwa gonadotropin-isohora imisemburo (GnRH) agoniste. Muri iyi nyandiko, tuzibanda ku mikoreshereze yayo mu kuvura kanseri ya prostate na kanseri y'ibere.

Kuvura Kanseri ya Prostate:
Leuprorelin ikunze gukoreshwa mu kuvura kanseri ya prostate yateye imbere. Irakora mukugabanya urwego rwa testosterone ikorwa na testicles. Ingirabuzimafatizo za kanseri ya prostate ziterwa na testosterone kugirango ikure, bityo kugabanya urwego rwayo bishobora kugabanya kanseri cyangwa kugabanya imikurire yayo. Ubuyobozi bwa leuprorelin bufasha gucunga ibimenyetso bifitanye isano na kanseri ya prostate kandi bikazamura imibereho yumurwayi.

Kuvura Kanseri y'ibere:
Leuprorelin ikoreshwa kandi mu kuvura ubwoko bumwe na bumwe bwa kanseri y'ibere. Ikoreshwa cyane cyane mugihe ingirabuzimafatizo za kanseri zifite reseptor ya estrogene (ER positif) kandi umurwayi akaba ataranyuze mu gucura. Leuprorelin igabanya urugero rwa estrogene mu mubiri ihagarika umusaruro wayo muri ovaries. Ibi ni ingenzi cyane kuko urugero rwa estrogene rushobora guteza imbere imikurire ya kanseri y'ibere. Leuprorelin irashobora gutangwa wenyine cyangwa ifatanije nubundi buryo bwo kuvura imisemburo kugirango kanseri ibere neza.


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Hagati y'ubwangavu bukuru:

Urushinge rwa Leuprorelin, ruzwi ku izina rya Lupron Depot-PED, rukoreshwa mu bana bafite imyaka 2 nayirenga mu kuvura ubwangavu bwibanze (CPP). CPP nuburyo abakobwa (mubisanzwe barengeje imyaka 8) nabahungu (mubisanzwe barengeje imyaka 9) binjira mubugimbi imburagihe. Leuprorelin ifasha kugenzura igihe cyubwangavu idindiza imikurire yamagufwa yihuse niterambere ryimiterere yimibonano mpuzabitsina ijyanye na CPP.


Ibindi bikoreshwa mu mavuriro:

Gutera Leuprorelin, bizwi kandi ku izina rya Lupron Depot, bikoreshwa mu kuvura endometriose na anemia biterwa na fibroide nyababyeyi. Ikora igabanya urugero rwa hormone zimwe na zimwe mu mubiri, itanga uburuhukiro bwibimenyetso nkububabare, imihango iremereye cyangwa idasanzwe, na anemia. Byongeye kandi, leuprorelin irashobora gukoreshwa nkubuvuzi mbere yubuvuzi mbere yo kwandura endometrale, kuko inanura endometrium, igabanya indurwe, kandi ikorohereza uburyo bwo kubaga.


Imiti ya farumasi:
Leuprorelin acetate ntabwo ikora neza iyo ifashwe kumunwa ahubwo igakoreshwa hakoreshejwe inshinge zidasanzwe cyangwa intanga. Nyuma yo guterwa inshuro imwe ya mg 3.75 mg, kwibumbira hamwe kwa plasma bigerwaho mugihe cyumunsi 1 kugeza 2, hamwe nurwego rwa 1 kugeza 2 ng / ml. Mu kuvura kanseri ya prostate, inshinge ya 3.75 mg itangwa buri byumweru 4 kugirango inshinge 3 zose hamwe kugirango igere kuri plasma ihagaze neza ya 0.1 kugeza 1 ng / ml. Leuprorelin ihindurwamo ibintu bine byangirika mu mubiri kandi bisohoka cyane binyuze mu mpyiko.

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Umwanzuro:
Leuprorelin, agoniste GnRH, nubuvuzi bwingirakamaro bwa hormone bukoreshwa mukuvura kanseri ya prostate na kanseri yamabere, hamwe nubwangavu bwibanze bwambere, endometriose, na anemia iterwa na fibroide nyababyeyi. Mugabanye urugero rwa testosterone cyangwa estrogene, leuprorelin ifasha kugenzura imikurire nibimenyetso bifitanye isano nibi bihe. Ubuyobozi bwa leuprorelin busaba kugenzurwa nubuvuzi no gukurikirana buri gihe kugirango bikore neza kandi bikemure ingaruka zose zishobora kubaho.

Wibuke kutwandikira kumpapuro zirambuye zo kohereza no kohereza, tuzatanga serivise zumwuga OEM / ODM.

Ibisobanuro

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