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Ifu ya Paroxetine Paroxetine Hydrochloride Ibikoresho bito Paroxetine Hcl

  • izina RY'IGICURUZWA Paroxetine
  • Kugaragara Ifu yera kugeza yera
  • URUBANZA No. 61869-08-7
  • Imiti yimiti C19H20FNO3
  • Uburemere bwa molekile 329.365403
  • Ingingo yo gushonga 118 - 125 C.
  • Ingingo yo guteka 451.674 ° C kuri 760 mmHg
  • Ubucucike 1.213
  • Ironderero 1.561

Ibisobanuro birambuye

Paroxetine isanzwe ikoreshwa nka hydrochloride cyangwa methanesulfonate.Hydrochloride ni umweru cyangwa yera, byoroshye gutanga ifu ya kristaline, byoroshye gushonga muri methanol, bigashonga gato muri Ethanol na methylene chloride, kandi bigashonga gato mumazi.Methanesulfonate ni ifu yera-yera. , impumuro nziza, gukomera mumazi> 1g / ml, gushonga ingingo 147 ~ 150 ℃.
Paroxetine ni imiti yingenzi ikoreshwa mu kuvura indwara zitandukanye zo mu mutwe, ni inkomoko ya fenylpiperidine na SSRI ishobora guhitamo kubuza abatwara 5-HT, guhagarika gufata 5-HT na membrane ya presinaptic, kuramba no kongera ingaruka. ya 5-HT, bityo ikabyara ingaruka zirwanya antidepressant. Igikorwa cyibanze ni ugukora nka antidepressant na anxiolytic agent muguhitamo guhitamo gufata serotonine mu bwonko.Serotonine ni neurotransmitter igira uruhare runini muguhindura imyumvire, amarangamutima, no guhangayika urwego.Mu guhagarika reuptake ya serotonine, Paroxetine ifasha kongera urugero rwa serotonine mu bwonko, bityo bigatuma umwuka uhinduka no kugabanya amaganya.

Paroxetine ikoreshwa kandi mu kuvura izindi ndwara z’ubuzima bwo mu mutwe nk’indwara idahwitse (OCD), ihungabana ry’imibereho, ihungabana ry’imibereho, hamwe n’ihungabana ry’ihungabana (PTSD) .Uburyo bwo gukora muri ibi bihe bisa n’ubwa uruhare mukuvura depression no guhangayika.Mu kongera urugero rwa serotonine mubwonko, Paroxetine ifasha kugabanya ibimenyetso bifitanye isano niyi ndwara.


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Ikoreshwa rya Paroxetine rikubiyemo ibintu byinshi byubuzima bwo mu mutwe, bituma biba imiti itandukanye kandi ifite agaciro.Nkuko imiti igabanya ubukana, Paroxetine ikoreshwa mu kugabanya ibimenyetso by’indwara ikomeye yo kwiheba, harimo umubabaro uhoraho, gutakaza inyungu mu bikorwa bisanzwe, impinduka mu ubushake cyangwa uburemere, guhungabana ibitotsi, no kumva ko nta gaciro ufite cyangwa kwicira urubanza. Mu kuvura indwara ziterwa no guhangayika, Paroxetine igira akamaro mu kugabanya ibimenyetso by’impungenge rusange, guhangayikishwa n’imibereho, hamwe n’ihungabana ry’ubwoba.Bifasha kugabanya impungenge zikabije, gutinya ibibazo by’imibereho. , n'ibitero by'ubwoba, bituma abantu bongera kugenzura amarangamutima yabo n'imikorere ya buri munsi.


Ku barwayi barwaye OCD, Paroxetine igira uruhare runini mugucunga imitekerereze n’agahato bibangamira ubuzima bwabo bwa buri munsi.Mu guhindura urugero rwa serotonine, Paroxetine ifasha kugabanya inshuro nuburemere bwibitekerezo bikabije ndetse nimyitwarire ihatira, bigatuma abantu bishora mubikorwa byabo bya buri munsi ibikorwa neza.Ikindi kandi, Paroxetine nayo ikoreshwa mukuvura PTSD, aho ifasha mukugabanya ibimenyetso bibabaza bifitanye isano nubunararibonye, ​​nkibitekerezo byinjira, inzozi mbi, hypervigilance, hamwe nimyitwarire yo kwirinda. Byongeye kandi, Paroxetine ikoreshwa hanze ya label. mugucunga ibindi bihe nka disphoric disorder (PMDD), ibimenyetso bya vasomotor bijyana no gucura, hamwe na syndromes zitandukanye. Izi porogaramu zitandukanye zerekana akamaro ka Paroxetine mugukemura ibibazo byinshi byubuzima bwo mumutwe.

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