Rosuvastatin antilipemic agent Rosuvastatin togafitia le dyslipidemia
Fa'amatalaga Auiliili
O le Rosuvastatin e taofia ai le enzyme hydroxymethylglutaryl-CoA reductase i le ate, lea e faʻaitiitia ai le faʻaogaina o le cholesterol ma faʻaititia ai le maualuga o le cholesterol ma le triglyceride. E le gata i lea, o le Rosuvastatin e faʻateleina ai le faʻaogaina o le ate ma malepelepe o le lipoprotein cholesterol maualalo (LDL-C), ae faʻateleina foi le maualuga o le lipoprotein cholesterol (HDL-C). I le faʻaopopoga i ona aʻafiaga e faʻaitiitia ai le lipid, o le Rosuvastatin ua faʻaalia e maua ai le anti-atherosclerotic, anti-inflammatory, antioxidant, faʻamautu o le plaque, ma faʻaleleia galuega endothelial.
O le Rosuvastatin e gaosia e ala i le faʻafefeteina o le Aspergillus terreus poʻo le faʻaogaina o vailaʻau. O le taimi lava e faʻaaogaina ai, e matua faʻafefeteina i le ate ma liua i ni metabolites eseese, e aofia ai metabolites malosi e taofia ai le HMG-CoA reductase. O le vailaʻau ma ona metabolites e faʻaulu muamua i feces, faʻatasi ai ma sina vaega itiiti e alu i le urine.