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Telmisartan Zviri nani antihypertensive Kudzivirira renal

Reference mutengo: USD 0.2-0.8/g

  • Product Name Telmisartan
  • CAS Nha. 144701-48-4
  • MF C33H30N4O2
  • MW 514.629
  • EINECS 1592732-453-0

Tsanangudzo Yakadzama

Telmisartan, inozivikanwawo seTimosartan, inova yeropa-inodzikisa BP yakarongedzwa seyakasiyana angiotensin II receptor (AT1-mhando) antagonist. Inoshandiswa zvakanyanya mukurapa yakakosha hypertension, ichipa zvakati wandei zvakanakira pane mamwe antihypertensive mishonga. Ichi chinyorwa chine chinangwa chekupa tarisiro yakazara yemabhenefiti eTelmisartan uye zvakakosha kufunga nezvekushandiswa kwayo.

Zvakanakira zveTelmisartan:

Zvirinani antihypertensive effect:
Telmisartan inowanzoshandiswa mumutsara wekutanga antihypertensive mushonga nekuda kwekunyanya kushanda kwayo. Semupikisi wemhando yeAT1, inodzivirira kuita kweangiotensin, zvichikonzera kudzikiswa kwakanyanya kweropa. Telmisartan inoratidza dhigirii repamusoro rekutsanangurwa kana ichienzaniswa nemamwe masartan, ichiibvumira kupinda zviri nyore mumasero membranes uye kunanga maseru chaiwo. Izvi zvinosimudzira mhedzisiro yayo yeantihypertensive, zvichikonzera kudzikira kwakanyanya muropa. Pamusoro pezvo, Telmisartan ine hafu yehupenyu hwakareba, inochengetedza uye inoshanda yekudzora kweropa.

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Kudzivirirwa kwemoyo uye cerebral midziyo:

Telmisartan inomira pachena seyo yega sartan-semushonga unobvumidzwa neFDA kune yayo yemoyo uye cerebrovascular inodzivirira zvivakwa. Inoratidza kukwanisa kudzoreredza kuruboshwe ventricular hypertrophy uye inokurudzirwa kune varwere vane hypertension inoperekedzwa nekuruboshwe ventricular hypertrophy, kushaya simba kwemoyo, kana coronary artery chirwere. Pamusoro peiyo BP-kudzikisa mhedzisiro, Telmisartan inoderedza kukuvara kwemoyo uye cerebrovascular. Inonyanya kubatsira kune vanhu vakambosangana nesitiroko kana cardiac infarction.

Kudzivirira renal function:

Imwe bhenefiti yeTelmisartan ndeye kunaka kwayo kukanganisa basa retsvo. Sezvo Telmisartan ichiita hepatic metabolism uye inoburitswa mubile, ine zvishoma zvinokanganisa basa retsvo. Uyezve, Telmisartan yakawanikwa ichideredza proteinuria, nekudaro ichichengetedza basa retsvo. Inonyanya kukosha kune varwere vane hypertension uye comorbid mamiriro akadai seshuga nephropathy, microalbuminuria, proteinuria, kana nyoro kusvika pakati nepakati renal insufficiency.

Kuvandudzwa kwe insulin kuramba:

Telmisartan yakaratidza mhedzisiro yakanaka paglucose metabolism uye insulin kuramba. Ichi chimiro chinoita kuti ive sarudzo yakakodzera kune varwere vane hypertension uye chirwere cheshuga mellitus, sezvo inogona kubatsira kuvandudza insulin senitivity uye kudzora glucose.


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Telmisartan, chaiyo angiotensin II receptor (AT1-mhando) anopikisa, inopa zvakati wandei zvakanakira mukurapa kwakakosha hypertension. Izvo zviri nani antihypertensive effect, kuchengetedzwa kwemidziyo yemwoyo uye cerebral, kuchengetedza renal basa, uye kuvandudzwa kwe insulin resistance inoita kuti ive sarudzo inokosha mukugadzirisa hypertension uye mamiriro akabatanidzwa. Nekudaro, zvakakosha kutevedzera nhungamiro inokurudzirwa maererano nenguva yemishonga, kutonga kwedosi, uye kugara uchitarisa kuti uve nechokwadi chekushanda uye kuchengetedzeka. Kuonana nenyanzvi yehutano inogara ichirairwa kuti uwane zano remunhu uye nhungamiro maererano nekushandiswa kweTelmisartan kana chero mushonga.

Tsanangudzo

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