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Leuprorelin Hormone Therapy ee Kansarka qanjirka 'prostate' iyo naasaha

Qiimaha tixraaca: USD 30-100

  • Magaca alaabta Leuprorelin
  • CAS Maya. 53714-56-0
  • Cufnaanta 1.44
  • barta dhalaalaysa 150-155°C
  • Barta karkarinta 1720.5°C at 760mmHg
  • MF C59H84N16O12
  • MW 1269.473
  • Tilmaanta refractive 1.681
  • Barta toosan 994.3°C

Sharaxaad faahfaahsan

Leuprorelin, oo sidoo kale loo yaqaan Lupron ama Prostap, waa daawaynta hoormoonka ee loo isticmaalo daaweynta qanjirka 'prostate' iyo kansarka naasaha. Waxay ka tirsan tahay koox dawooyin ah oo loo yaqaanno gonadotropin-sii daynta hormoonnada (GnRH) agonists. Qormadan, waxaan diiradda saari doonaa isticmaalkeeda daaweynta kansarka qanjirka 'prostate' iyo kansarka naasaha.

Daaweynta Kansarka qanjirka 'prostate':
Leuprorelin waxaa badanaa loo isticmaalaa in lagu daaweeyo kansarka qanjirka 'prostate'. Waxay u shaqeysaa iyada oo hoos u dhigaysa heerka testosterone ee ay soo saaraan xiniinyaha. Unugyada kansarka qanjirka 'prostate' waxay ku tiirsan yihiin testosterone si ay u koraan, markaa hoos u dhigista heerarkeeda waxay hoos u dhigi kartaa kansarka ama waxay hoos u dhigi kartaa koritaankeeda. Maamulka leuprorelin wuxuu caawiyaa maaraynta calaamadaha la xidhiidha kansarka qanjirka 'prostate' ee sare u kacay waxayna wanaajisaa tayada nolosha bukaanka.

Daaweynta Kansarka Naasaha:
Leuprorelin waxa kale oo loo isticmaalaa daawaynta noocyo ka mid ah kansarka naasaha. Waxaa si gaar ah loo isticmaalaa xaaladaha ay unugyada kansarku leeyihiin estrogen reseptors (ER positive) oo bukaanku aanu soo marin menopause. Leuprorelin wuxuu yareeyaa heerka estrogen ee jirka isagoo xakameynaya wax soo saarkiisa ugxan-sidaha. Tani waa muhiim sababtoo ah heerarka sare ee estrogen waxay kor u qaadi karaan koritaanka unugyada kansarka naasaha. Leuprorelin waxaa la qaadan karaa kaligiis ama lagu daro daawaynta hoormoonka kale si loo maareeyo kansarka naasaha.


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Barbaarinta Precocious:

Cirbadka Leuprorelin, oo loo yaqaan Lupron Depot-PED, ayaa loo isticmaalaa carruurta da'doodu tahay 2 sano iyo ka weyn si loogu daweeyo baaluqnimada dhexe ee precocious (CPP). CPP waa xaalad ay habluhu (badanaa ka yar yihiin 8 sano) iyo wiilasha (badanaa ka yar da'da 9 sano) ay galaan qaangaar degdeg ah. Leuprorelin waxay caawisaa habaynta wakhtiga qaan-gaarnimada iyadoo hoos u dhigaysa koritaanka degdega ah ee lafaha iyo horumarinta sifooyinka galmada ee la xidhiidha CPP.


Isticmaalka Caafimaad ee Kale:

Cirbadda Leuprorelin, oo sidoo kale loo yaqaan Lupron Depot, ayaa loo adeegsadaa daaweynta endometriosis iyo dhiig-yaraan ay keento fibroids uterineine. Waxay u shaqeysaa iyadoo hoos u dhigaysa heerarka hormoonnada qaarkood ee jirka, iyadoo bixisa nafis calaamadaha sida xanuunka, caadada culus ama aan joogtada ahayn, iyo dhiig-yaraan. Intaa waxaa dheer, leuprorelin waxaa loo isticmaali karaa sidii hore daaweyn caafimaad ka hor inta aan la soo saarin endometrial, maadaama ay khafiifiso endometrium, yareyso bararka, waxayna fududeysaa habka qalliinka.


Farmashiyaha:
Leuprorelin acetate ma aha mid wax ku ool ah marka afka laga qaato waxaana taas bedelkeeda lagu maamulaa cirbadeynta muruqa hoose ama gudaha. Ka dib hal cirbad oo subcutaneous ah oo ah 3.75 mg, diirada ugu sarreysa balaasmaha ayaa lagu gaaraa 1 ilaa 2 maalmood gudahood, oo leh heerar 1 ilaa 2 ng/ml. Daawaynta kansarka qanjirka 'prostate', cirbadeynta subcutaneous ee 3.75 mg ayaa la bixiyaa 4tii usbuucba mar wadarta guud ee 3 irbadood si loo gaaro xajmiyada balasmaha ee 0.1 ilaa 1 ng/ml. Leuprorelin waxa loo qaybiyaa afar badeecooyin nabaad-guur ah oo jidhka ku jira waxana laga soo saaraa kelyaha.

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Gabagabo:
Leuprorelin, GnRH agonist, waa daawaynta hoormoonka qiimaha leh ee loo isticmaalo daawaynta qanjirka 'prostate' iyo kansarka naasaha, iyo sidoo kale baaluqnimada dhexe ee precocious, endometriosis, iyo dhiig-yaraan ay keento fibroids uterineine. Iyada oo la yareeyo heerarka testosterone ama estrogen, leuprorelin waxay ka caawisaa xakameynta korriinka iyo calaamadaha la xiriira xaaladahan. Maamulka leuprorelin wuxuu u baahan yahay kormeer caafimaad iyo kormeer joogto ah si loo hubiyo waxtarkeeda oo loo maareeyo waxyeelo kasta oo iman karta.

Xusuusnow inaad nala soo xiriirto baakadaha faahfaahsan iyo foomamka rarida, waxaan ku siin doonaa adeegyo xirfadeed OEM/ODM hagaajinta.

Tilmaamid

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