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Telmisartan Betere antihypertensive Ho sireletsa renal

Theko ea litšupiso: USD 0.2-0.8/g

  • Lebitso la Sehlahiswa Telmisartan
  • Nomoro ea CAS. 144701-48-4
  • MF C33H30N4O2
  • MW 514.629
  • EINECS 1592732-453-0

Tlhaloso e Felletseng

Telmisartan, eo hape e tsejoang e le Timosartan, ke sethethefatsi se secha se theolang khatello ea mali se thathamisitsoeng e le mohanyetsi ea itseng oa angiotensin II receptor (mofuta oa AT1). E sebelisoa haholo kalafong ea khatello ea mali ea bohlokoa, e fanang ka melemo e mengata ho feta litlhare tse ling tsa antihypertensive. Moqoqo ona o ikemiselitse ho fana ka kakaretso e felletseng ea melemo ea Telmisartan le lintlha tsa bohlokoa bakeng sa ts'ebeliso ea eona.

Lintho tse molemo tsa Telmisartan:

Phello e ntle ea antihypertensive:
Telmisartan ke setlhare sa pele sa antihypertensive se laetsoeng ka lebaka la katleho ea sona e phahameng. Joaloka mohanyetsi oa mofuta oa AT1, e thibela ketso ea angiotensin, e bakang phokotso e kholo ea khatello ea mali. Telmisartan e bonts'a maemo a holimo ha a bapisoa le li-sartan tse ling, e e lumellang hore e kene ka har'a lisele le ho shebana le lisele tse itseng. Sebopeho sena se ntlafatsa litlamorao tsa eona tsa antihypertensive, se lebisang ho fokotseha ho hoholo ha khatello ea mali. Ntle le moo, Telmisartan e na le halofo ea bophelo bo bolelele, e netefatsa taolo e tsitsitseng le e sebetsang ea khatello ea mali.

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Tšireletso ea methapo ea pelo le ea boko:

Telmisartan e hlahella e le eona feela sethethefatsi se kang sartan se amohetsoeng ke FDA bakeng sa thepa ea eona ea ts'ireletso ea pelo le cerebrovascular. E bontša bokhoni ba ho khutlisa hypertrophy ea ventricular e ka morao 'me e khothalletsoa bakuli ba nang le khatello ea kelello e tsamaeang le le letšehali ventricular hypertrophy, ho se sebetse ha pelo, kapa lefu la methapo ea mali. Ntle le litlamorao tsa eona tsa ho theola khatello ea mali, Telmisartan e fokotsa tšenyo ea pelo le methapo ea mali. E bohlokoa haholo ho batho ba nang le stroke kapa infarction ea pelo.

Ho sireletsa mosebetsi oa renal:

Molemo o mong oa Telmisartan ke phello e ntle mosebetsing oa renal. Kaha Telmisartan e kena metabolism ea sebete 'me e ntšoa ka bile, e na le phello e fokolang mosebetsing oa renal. Ho feta moo, Telmisartan e fumanoe e fokotsa proteinuria, ka hona e sireletsa ts'ebetso ea renal. E bohlokoa haholo ho bakuli ba nang le khatello ea mali le maemo a comorbid joalo ka nephropathy ea lefu la tsoekere, microalbuminuria, proteinuria, kapa ho se sebetse hantle hoa renal ha bobebe ho isa bohareng.

Ho ntlafatsa ho hanyetsa insulin:

Telmisartan e bonts'itse litlamorao tse ntle ho metabolism ea tsoekere le ho hanyetsa insulin. Tšobotsi ena e etsa hore e be khetho e nepahetseng bakeng sa bakuli ba nang le khatello ea mali le lefu la tsoekere, kaha e ka thusa ho ntlafatsa kutloisiso ea insulin le taolo ea tsoekere.


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Telmisartan, mohanyetsi ea itseng oa angiotensin II receptor (AT1-mofuta) e fana ka melemo e mengata kalafong ea khatello ea mali ea bohlokoa. Phello ea eona e ntle ea antihypertensive, ts'ireletso ea methapo ea pelo le ea boko, ho boloka ts'ebetso ea renal, le ntlafatso ea ho hanyetsa insulin ho etsa khetho ea bohlokoa ho laola khatello ea mali le maemo a amanang. Leha ho le joalo, ho bohlokoa ho latela litataiso tse khothaletsoang mabapi le nako ea meriana, taolo ea litekanyetso, le ho beha leihlo khafetsa ho netefatsa ts'ebetso e nepahetseng le polokeho. Ho buisana le setsebi sa bophelo bo botle ho lula ho eletsoa bakeng sa likeletso le tataiso ea motho ka mong mabapi le ts'ebeliso ea Telmisartan kapa moriana ofe kapa ofe.

Tlhaloso

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