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I-Dapoxetine powder tablet I-Dapoxetine I-Ejaculation yangaphambi kwexesha kuMadoda
Inkcazo eneenkcukacha
I-Dapoxetine, i-CAS No. 119356-77-3, kunye ne-molecular formula C21H23NO, iyeza elisetyenziselwa unyango lwe-ejaculation ngaphambi kwexesha kumadoda. Ibonakala ngathi ngumgubo wekristale omhlophe ukuya kumhlophe, kwaye awunavumba. I-Dapoxetine ine-solubility encinci emanzini.
I-Dapoxetine powder luhlobo olutsha lwe-SSRI ekhawulezayo kunye nesiqingatha sobomi obufutshane. Yinto ekhethiweyo ye-serotonin reuptake inhibitor (SSRI). Lichiza elisetyenziselwa ukunyanga ukuphuma kwangaphambi kwexesha kumadoda aneminyaka eyi-16 ukuya kuma-84 ubudala.
Kwisigaba sesi-II sophando lobungqina bobungqina olwenziwa yiPPD, i-dapoxetine ibonise ukwanda kwezibalo kwi-ejaculatory latency xa kuthelekiswa ne-placebo. Idosi eninzi.
I-Dapoxetine (INN, i-brand name Priligy), ifom ye-dosage esetyenziswa ngokuqhelekileyo iipilisi, sikwaxhasa ii-capsules ezenziwe ngokwezifiso. Ekuqaleni yaphuhliswa njenge-antidepressant, kamva yafunyanwa ukuba nayo inokusebenza kakuhle ekuphatheni i-ejaculation ngaphambi kwexesha (PE). Ngoku ithathwa njengonyango olusebenzayo lokuphuma kwangaphambi kwexesha emadodeni. I-Dapoxetine inokwandisa ixesha lokwabelana ngesondo kumadoda, ngaloo ndlela iphucula umgangatho wobomi babo besondo. I-Dapoxetine iguqula i-nerve conduction ngokuvimbela ukubuyiswa kwakhona kwe-serotonin, ngaloo ndlela inyusa ukuxinwa kwe-serotonin kwii-synapses. Esi senzo sivumela i-dapoxetine ukuba yandise ixesha lokwabelana ngesondo, ngaloo ndlela inceda amadoda ahlupheke kwiingxaki ze-ejaculation ngaphambi kwexesha. I-dose yonyango ye-dapoxetine idla ngokuba yi-30mg okanye i-60mg, enokuthi ihlengahlengiswe ngokwemeko yangempela yesigulane. Ifunxwa ngokukhawuleza emva kokulawulwa komlomo kwaye ithatha malunga neeyure ezingama-1-2 ukufikelela kwincopho yoxinaniso lweplasma. Ubomi besiqingatha se-dapoxetine malunga neeyure ze-1-2, oku kuthetha ukuba i-metabolized kwaye ikhutshwe ngokukhawuleza emzimbeni. Kwizigulane ezininzi, ukusetyenziswa kwe-dapoxetine kukhuselekile, kodwa ezinye iimpendulo ezimbi zinokuthi zenzeke, kubandakanywa intloko, isicathulo, ukulala, ukukhathala, njl. Ngaphambi kokuba uqale i-dapoxetine, kufuneka uthethe nodokotela wakho ukuqinisekisa ukuba akukho mngcipheko wokusebenzisana nezinye amayeza okanye iimeko zonyango ezikhoyo.