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I-Tirzepatide Dual GLP-1 kunye ne-GIP Receptor Agonist yoLawulo lobunzima kunye noLawulo lweGlycemic

Ixabiso lokubhekisela: USD 300-600/g

  • Igama lemveliso Tirzepatide
  • Inombolo yeCAS. 2023788-19-2
  • MF C225H348N48O68
  • MW 4813.45

Inkcazo eneenkcukacha

I-Tirzepatide liyeza elinoveli elisetyenziselwa ukulawula ubunzima bexesha elide kwizigulana ezityebileyo ngokutyeba kwabantu abadala okanye i-comorbidities ezinxulumene nobunzima. I-agonist exhomekeke kwi-glucose ye-glucagon polypeptide (GIP) kunye ne-glucagon-like peptide-1 (GLP-1) receptors. Ivunywe yi-FDA ngo-2022, i-tirzepatide idibanisa iziphumo ze-enteric proinsulins kwi-molecule enye, iphucula ukukhutshwa kwe-insulin kunye nokunciphisa amanqanaba eglucagon. Eli nqaku liphonononga indlela yokusebenza, ukusebenza kweklinikhi, kunye neprofayili yokhuseleko lwe-tirzepatide njengonyango lokuncedisa ukunciphisa umzimba kunye nokuphucula ulawulo lwe-glycemic kwizigulane ezine-2 yeswekile.

I. Ukuqonda iTirzepatide:
A. I-agonist exhomekeke kwi-Glucose ye-GIP kunye ne-GLP-1 receptors
B. Inkqubo yesenzo: ukuphucula isigaba soku-I kunye nesigaba II se-insulin secretion, ukunciphisa amanqanaba eglucagon

II. Usetyenziso lweKlinikhi kunye neMvume ye-FDA:
A. Isalathiso: Ukulawulwa kwexesha elide lobunzima kwizigulane ezityebileyo kunye nokutyeba kwabantu abadala okanye ubunzima obunxulumene nobunzima
B. Unyango olongezelelweyo lokuphucula ulawulo lwe-glycemic kubantu abadala abanesifo sikashukela sohlobo lwe-2
C. Ukwamkelwa kwe-FDA kunye nokuthengiswa ngu-Eli Lilly ngo-2022

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III. Ukusebenza kakuhle kuLawulo lobunzima:

A. Ukusebenza ngokuthelekisayo:

Ipesenti yokulahleka kwesisindo: Idosi ephantsi (5mg), idosi ephakathi (10mg), kunye nedosi ephezulu (15mg) amaqela

Umyinge weepesenti zokulahleka kobunzima kumaqela ahlukeneyo edosi

Ukuthelekisa neqela le-placebo

Ipesenti yezifundo ezifumana ukwehla kobunzima ngaphezu kwe-20%

B. Iprofayile yokhuseleko: Ukuphindaphinda kweempendulo ezingalunganga xa kuthelekiswa neqela le-placebo

C. Ukuthelekiswa namanye amayeza okunciphisa umzimba:

I-Orlistat (i-over-the-counter): Umahluko kwiipesenti zokulahlekelwa kwesisindo


IV. Indlela yoLawulo lweGlycemic kunye nokuLahla kobunzima:

A. Ukusetyenziswa kwe-GLP-1 kunye ne-GIP receptors

B. Ukunciphisa ukutya kunye nokunciphisa ukutya okutyayo



17158639023143ie


I-Tirzepatide, njenge-GLP-1 emibini kunye ne-GIP receptor agonist, ibonelela ngolawulo olusebenzayo lobunzima kunye nokuphuculwa kokulawulwa kwe-glycemic kwizigulane ezityebileyo kunye nokukhuluphala kwabantu abadala okanye ubunzima obunxulumene nobunzima, kunye nabantu abanesifo sikashukela sohlobo lwe-2. Indlela yokusebenza exhomekeke kwiglucose inyusa ukukhutshwa kwe-insulin kunye nokunciphisa amanqanaba eglucagon. Ngeepesenti ezibalulekileyo zokulahlekelwa kwesisindo kunye neprofayili ekhuselekileyo yokhuseleko, i-tirzepatide ivelele njengamayeza anamandla okulawula ubunzima bexesha elide. Uphando olongezelelweyo kunye nezifundo zeklinikhi ziyakuqhuba ziphonononga iinzuzo ezinokuthi zibekho kunye nokusetyenziswa kweli chiza lithembisayo.
Ukuze unikeze amava okurhweba angcono, sinokwenza i-capsule kunye neemveliso zolwelo, ngokweemfuno zakho zezithako.
Sinokwenza ngokwezifiso umthamo: 500mg / capsule, 550mg / capsule, 600mg / capsule.
Siyakwazi ukwenza ngokwezifiso ukupakishwa: 60 caps / ibhotile, 90 caps / ibhotile, 120 caps / ibhotile.
Sinokwenza ngokwezifiso iigobolondo ze-capsule kunye nemibala: iigobolondo ze-capsule yezityalo, iigobolondo ze-gelatin capsule.

Inkcazo

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