Incazelo Eningiliziwe
I-Tadalafil iyi-crystalline powder emhlophe kuya kokumhlophe. Ayincibiliki emanzini, ibonisa ukuncibilika kancane, futhi incibilika kancane otshwaleni.Into ehlanzekile ayinaphunga futhi ayinambitheki, iveza njengempushana ecolekile, eyicrystalline.
Umsebenzi oyinhloko we-Tadalafil ukwelapha ukungasebenzi kahle kwe-erectile ngokwandisa ukugeleza kwegazi epipini ngesikhathi sokuvuselela ucansi.Ifeza lokhu ngokuvimbela i-enzyme phosphodiesterase uhlobo 5(PDE5), olubangela ukuwohloka kwe-cyclic guanosine monophosphate(cGMP) ku-corpus cavernosum. Ngokuvimbela i-PDE5, i-tadalafil ivumela i-vasodilation isikhathi eside kanye nokugeleza kwegazi okwandisiwe, okusiza amadoda ane-erectile dysfunction ukuze afinyelele futhi asekele ukuqhanyelwa.Ngokungafani neminye imithi ye-ED, i-tadalafil inesikhathi eside sokusebenza, nemiphumela ehlala njalo amahora angu-36, uthole igama lesidlaliso "iphilisi lempelasonto."
I-Tadalafil iboniswa ngokuyinhloko ekwelapheni i-erectile dysfunction (ED) kwabesilisa abadala. Itholakala ngendlela yethebhulethi ukuze iphathwe ngomlomo, ngemithamo esukela ku-2.5 mg kuya ku-20 mg, kuye ngezidingo zesiguli kanye nesimo eselashwayo. Umthamo wokuqala onconyiwe weziguli eziningi ngu-10 mg, othathwa ngaphambi kocansi okulindelekile, kanye nokudla noma ngaphandle kokudla. Umthamo ungalungiswa ngokusekelwe ekubekezeleleni komuntu ngamunye kanye nokuphendula.Ngaphezu kokusetshenziswa kwayo kwe-erectile dysfunction, i-tadalafil iphinde ivunyelwe ukwelashwa kwezibonakaliso nezimpawu ze-benign prostatic hyperplasia(BPH), isimo esibonakala nge-prostate gland ekhulisiwe. Lapho i-BPH ihambisana nokungasebenzi kahle kwe-erectile, i-tadalafil inganikeza inzuzo ekabili ngokubhekana nezimo zombili ngesikhathi esisodwa.
Ngaphezu kwalokho, i-tadalafil isetshenziselwa ukuphatha i-pulmonary arterial hypertension(PAH) kokubili amadoda nabesifazane. Kulolu hlelo lokusebenza, kusiza ukuthuthukisa amandla okuzivocavoca futhi kubambezele ukuwohloka komtholampilo kwalesi sifo.
Sengiphetha, i-tadalafil iyi-crystalline powder emhlophe ukuya kokumhlophe enokuncibilika okulinganiselwe, ngokuyinhloko isetshenziselwa ukwelapha ukungasebenzi kahle kwe-erectile, i-benign prostatic hyperplasia, kanye nomfutho wegazi ophakeme we-pulmonary arterial. Njenge-PDE5 inhibitor, yenza kube lula ukugeleza kwegazi ezindaweni ezithile zomzimba, ikakhulukazi umthondo, okwenza kube ngcono ukusebenza kwe-erectile. Ukwengeza, ubude bayo besenzo buyenza ihluke kweminye imithi ekilasini layo, inikeze ukuguquguquka nokuzenzakalelayo kubantu abafuna ukwelashwa kwe-ED.
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