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I-YK-11 I-SARM Enamandla Yokwakhiwa Kwemisipha, Ukuzuza Amandla, kanye Ne-Myostatin Inhibition

Intengo Yereferensi:USD 40-150/g

  • Igama Lomkhiqizo YK11
  • Inombolo ye-CAS. 431579-34-9
  • MF I-C25H34O6
  • MW 430.541
  • Ukuminyana 1.2±0.1 g/cm3
  • Iphuzu elibilayo 564.4±50.0 °C ku-760 mmHg

Incazelo Eningiliziwe

I-YK-11 iyi-modulator ye-androgen receptor (SARM) ekhethiwe ethole ukuthandwa emphakathini wokwakha umzimba. Kuyaziwa ngekhono layo lokunamathisela ngokukhetha kuma-androgen receptors athile, ukuvimbela umsebenzi we-myostatin nokukhuthaza ukukhula kwemisipha. Lesi sihloko sihlola ukuthi i-YK-11 isebenza kanjani, izinzuzo zayo ekwakheni umzimba, ukusetshenziswa okunconyiwe, kanye nokusebenza kwayo ekwakhiweni kwemisipha (bulking) nokulahlekelwa kwamafutha (ukusika).

I. Ukuqonda i-YK-11:
A. YK-11 njenge-SARM ene-androgen receptor ebophayo
B. Ihlukile kuma-anabolic steroids, aqondise ama-receptors athile
C. Ukuvinjelwa kwephrotheni ye-myostatin ukukhuthaza ukukhula kwemisipha
D. Isakhiwo esifanayo sejometri kuma-anabolic steroids

II. Indlela Yesenzo:
A. Indima ye-Myostatin ekuvimbeleni ukukhula kwemisipha
B. Indima ye-Follistatin ekuzuzweni kwemisipha namandla
Ikhono le-C. YK-11 lokwehlisa amazinga e-myostatin nokwandisa i-follistatin
D. Ukungeniswa kwamangqamuzana emisipha ukuze kukhiqizwe i-follistatin eyengeziwe

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III. Izinzuzo ze-YK-11:

A. Isisindo somzimba esithuthukisiwe namandla azuzayo

B. Amathuba okudlula imikhawulo yokukhula kwemisipha yofuzo

C. Ukuthuthukiswa kokuqina kwamathambo nokukhula kwamangqamuzana amathambo

D. Ukufana ne-testosterone ekukhuthazeni ukukhula kwemisipha


IV. Ukusetshenziswa kwe-YK-11 Ekwakhiweni Komzimba:

A. Ifanele ukunqwabelana, ukusika, nomjikelezo wokubuyisela

B. Umthamo onconyiwe: 10-15 mg/day for mass building

C. Abasebenzisi bokuqala kufanele baqale ngama-SARM athambile

D. Ukungaguquguquki kokuqeqeshwa kanye nokudla okufanele kubalulekile


V. YK-11 Umjikelezo Nesilinganiso:

A. Ubude besikhathi esisebenzayo nesiphephile somjikelezo: 8 amaviki

B. Umthamo onconyiwe osuselwe kusisindo somzimba (10-15 mg/ngosuku)

C. Umthamo olondolozayo wabasebenzisi bokuqala noma ngesikhathi sokusika/ukubuyisela (5 mg/ngosuku)

D. PCT (Post Cycle Therapy) nge-Clomid (20 mg/day) amaviki angu-4


VI. I-YK-11 Yokwakha Imisipha (Ukugcwala Okuningi) Nokulahlekelwa Kwamafutha (Ukusika):

A. Ukuhlukahluka kwe-YK-11 kuzo zombili izinhloso

B. Isilinganiso esiphansi ngesikhathi sokulahlekelwa kwamafutha ukuze kugcinwe isisindo semisipha

C. Ukuhlola ukubekezelelana kanye nokukhuphuka kwethamo okungaba khona ekwakheni imisipha

D. Izinketho zesitaki nge-LGD 4033 ukuze uthole imiphumela ethuthukisiwe


Ngaphezu kwalokho, i-tadalafil isetshenziselwa ukuphatha i-pulmonary arterial hypertension(PAH) kokubili amadoda nabesifazane. Kulolu hlelo lokusebenza, kusiza ukuthuthukisa amandla okuzivocavoca futhi kubambezele ukuwohloka komtholampilo kwalesi sifo.

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I-YK-11 iyi-SARM enamandla enikeza izinzuzo ezibalulekile zokwakha imisipha, izinzuzo zamandla, kanye nokuvinjelwa kwe-myostatin. Ikhono layo lokukhomba ngokukhetha ama-androgen receptors kanye nokulawula amazinga e-myostatin kwenza kube inhlanganisela ebalulekile ekwakheni umzimba. Kungakhathaliseki ukuthi i-bulking noma ukusika, i-YK-11 ingafakwa emijikelezweni enedosi efanele kanye nobude besikhathi somjikelezo, ephelezelwa Ukwelashwa Komjikelezo Okufanele. Nakuba i-YK-11 isebenza kakhulu, kubalulekile ukubeka phambili ukuphepha futhi ulandele imihlahlandlela yokusetshenziswa enconyiwe ukuze wandise izinzuzo zayo.
Njengomphakeli ochwepheshe, singakwazi ukwenza ngokwezifiso i-capsule nemikhiqizo yoketshezi, ngokuya ngezidingo zakho zezithako.
Singakwazi ukwenza ngokwezifiso umthamo: 500mg/capsule, 550mg/capsule, 600mg/capsule.
Singakwazi ukwenza ngokwezifiso ukupakishwa: 60 caps / ibhodlela, 90 caps / ibhodlela, 120 caps / ibhodlela.
Singakwazi ukwenza ngokwezifiso amagobolondo we-capsule nemibala: amagobolondo e-capsule yezitshalo, amagobolondo we-gelatin capsule.

Ukucaciswa

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