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Linaclotide Ib Ntau Yam Peptide rau Cov Kabmob Plawv thiab Kev Noj Qab Haus Huv

  • Khoom npe Linaclotide
  • CAS Nr. 851199-59-2
  • MF C59H79N15O21S6
  • MW 1526.74 ib
  • Qhov tshwm sim Dawb lub zog
  • Acidity coefficient (pka) 3.05 ± 0.10 (Kev kwv yees)

Cov lus piav qhia ntxaws

Linaclotide, peptide agonist ntawm guanylate cyclase 2C, tau tshwm sim los ua qhov kev xaiv zoo tshaj plaws rau kev kho mob ntawm ntau yam plab hnyuv. Nrog nws cov khoom tshwj xeeb thiab cov txheej txheem ntawm kev ua, Linaclotide muaj ntau cov txiaj ntsig hauv kev tswj hwm plab hnyuv siab raum (IBS) thiab mob plab idiopathic constipation (CIC). Tsis tas li ntawd, nws muaj peev xwm txuas ntxiv mus rau kev txo qis ntawm plab zom mov, gastritis, plab ulcers, gastroesophageal reflux kab mob (GERD), thiab kev tiv thaiv thiab kho cov kab mob peptic.

Linaclotide rau cov kab mob hauv plab:
Linaclotide tau ua pov thawj tias muaj txiaj ntsig zoo hauv kev kho mob plab plob tsis so tswj nrog cem quav (IBS-C) thiab mob plab idiopathic constipation (CIC). Los ntawm kev ua kom cov kua dej hauv cov hnyuv thiab txhawb kev txav ntawm cov zaub mov los ntawm lub plab, Linaclotide pab txo cov tsos mob xws li tsam plab, mob plab, tsis xis nyob, straining, thiab kev xav ntawm lub plab zom mov tsis tiav. Nws lub peev xwm los txo qis kev ua haujlwm ntawm cov kab mob colonic sensory neurons txo qhov mob, thaum activating colonic motor neurons tsub kom cov leeg nqaij contraction thiab txhawb plab hnyuv.

Relieving plab hnyuv thiab gastritis:
Ntxiv nrog rau nws cov txiaj ntsig hauv kev tswj cov kab mob hauv plab, Linaclotide tau pom cov lus cog tseg hauv kev txo cov tsos mob ntawm plab hnyuv thiab gastritis. Los ntawm alleviating plab chim siab, mob, thiab tsam plab, Linaclotide capsules muab kev pab los ntawm kev xav tsis zoo. Tsis tas li ntawd, Linaclotide tuaj yeem txo qis hauv plab acid secretion thiab txo qhov tshwm sim ntawm gastric o, pab txhawb kev zom zaub mov zoo.

Kev kho mob plab ulcers:
Linaclotide capsules yog dav siv rau kev kho mob plab ulcers. Los ntawm inhibiting gastric acid secretion thiab txhawb txoj kev kho, Linaclotide pab kho cov kab mob plab. Nws kuj txo qhov kev pheej hmoo ntawm rwj rov tshwm sim thiab ua kom lub plab muaj peev xwm tiv thaiv. Cov khoom no ua rau Linaclotide yog ib qho kev xaiv zoo rau kev tswj thiab tiv thaiv kab mob plab.

Kev pab los ntawm Gastroesophageal Reflux Disease (GERD):
Linaclotide capsules tau pom tias muaj txiaj ntsig zoo hauv kev txo cov tsos mob cuam tshuam nrog tus kab mob gastroesophageal reflux. Mob plawv, mob hauv siab, thiab hnoos los ntawm cov kua qaub reflux tuaj yeem kho tau zoo nrog Linaclotide. Tsis tas li ntawd, Linaclotide pab kho cov kab mob hauv plab hnyuv, txo qhov mob, thiab tiv thaiv kev puas tsuaj ntxiv.

Kev Tiv Thaiv thiab Kev Kho Mob Peptic Ulcers:
Linaclotide capsules ua lub luag haujlwm tseem ceeb hauv kev tiv thaiv thiab kho kab mob peptic. Los ntawm inhibiting gastric acid secretion, Linaclotide txo qhov tshwm sim thiab rov tshwm sim ntawm rwj. Tsis tas li ntawd, nws txhawb kev kho rwj thiab ua kom cov txheej txheem kho mucosal, pab kom rov zoo tag nrho ntawm lub plab noj qab haus huv.

Kev pab los ntawm poob qab los ntawm Gastritis:
Linaclotide tau pom tias txo qis qab los noj mov cuam tshuam nrog gastritis. Itsanti-inflammatory zog pab txo lub plab o thiab txhim kho kev zom zaub mov ntawm lub plab. Raws li qhov tshwm sim, Linaclotide txhawb kev rov qab los ntawm kev qab los noj mov thiab nce kev noj zaub mov, hais txog qhov teeb meem ntawm kev poob qab los ntawm gastritis.

Kev tswj ntawm gastric acid ntau lawm:
Ib qho txiaj ntsig tseem ceeb ntawm Linaclotide yog nws lub peev xwm los tswj cov kua qaub hauv plab. Los ntawm kev txo qis hauv plab acid secretion, Linaclotide pab tswj cov kua qaub-puag ib puag ncig hauv plab. Qhov kev tswj hwm ntawm gastric acid ntau lawm tsis tsuas yog pab txhawb rau tag nrho cov plab hnyuv siab raum tab sis kuj tswj tau cov kab mob gastric acid xws li gastric ulcers thiab gastroesophageal reflux kab mob.

Tsis tas li ntawd, tadalafil yog siv los tswj pulmonary arterial hypertension (PAH) hauv cov txiv neej thiab poj niam. Hauv daim ntawv thov no, nws pab txhim kho kev tawm dag zog lub cev thiab ncua kev kho mob ntawm tus kab mob.

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Linaclotide, raws li kev tswj hwm peptide agonist ntawm guanylate cyclase 2C, muaj ntau yam txiaj ntsig rau kev kho mob plab hnyuv thiab plab hnyuv. Nws lub peev xwm los txo cov tsos mob ntawm kev chim siab plob tsis so tswj syndrome thiab mob idiopathic cem quav tau zoo tsim. Tsis tas li ntawd, Linaclotide qhia cov lus cog tseg hauv kev txo cov plab zom mov, gastritis, thiab kab mob gastroesophageal reflux. Nws tseem ua lub luag haujlwm tseem ceeb hauv kev tiv thaiv thiab kho mob plab thiab peptic ulcers. Thaum Linaclotide muab kev pab cuam tseem ceeb thiab txhawb txoj kev noj qab haus huv ntawm txoj hnyuv, nws yog ib qho tseem ceeb uas yuav tau sab laj nrog kws kho mob rau kev siv kom tsim nyog thiab kev coj noj coj ua.

Specification

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