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Paroxetine Powder Paroxetine Hydrochloride Raw Material Paroxetine Hcl

  • Lebitso la Sehlahiswa Paroxetine
  • Ponahalo Phofo e tšoeu ho isa ho bosoeu
  • Nomoro ea CAS. 61869-08-7
  • Foromo ea Lik'hemik'hale Setšoantšo sa C19H20FNO3
  • Boima ba molek'hule 329.365403
  • Sebaka se qhibilihang 118 - 125 C
  • Ntho e belang 451.674 °C ho 760 mmHg
  • Botenya 1.213
  • Lenane la refractive 1.561

Tlhaloso e Felletseng

Paroxetine e atisa ho sebelisoa e le hydrochloride ea eona kapa methanesulfonate.Hydrochloride e tšoeu kapa ha e tšoeu, e bonolo ho kristale phofo, e qhibiliha habonolo ka methanol, e qhibiliha hanyenyane ka ethanol e feletseng le methylene chloride, 'me e qhibiliha hanyenyane metsing. ,ha e na monko, ho qhibiliha ka metsing>1g/ml, ntlha e qhibilihisang 147~150℃.
Paroxetine ke meriana ea bohlokoa e sebelisetsoang ho phekola maemo a sa tšoaneng a bophelo bo botle ba kelello, ke motsoako oa phenylpiperidine le SSRI e ka thibelang sepalangoang sa 5-HT, thibela reuptake ea 5-HT ka lesela la presynaptic, lelefatsa le ho eketsa phello. ea 5-HT, ka hona e hlahisa phello e thibelang ho imeloa kelellong. Mosebetsi oa eona o ka sehloohong ke ho sebetsa e le sethethefatsi se thibelang ho tepella maikutlo le ho tšoenyeha ka ho thibela ka mokhoa o ikhethileng ho tsosolosoa ha serotonin bokong.Serotonin ke neurotransmitter e bapalang karolo ea bohlokoa ho laola maikutlo, maikutlo le matšoenyeho. Ka ho thibela ho tsosolosoa ha serotonin, Paroxetine e thusa ho eketsa maemo a serotonin bokong, ka tsela eo ho ntlafatsa maikutlo le ho fokotsa ho tšoenyeha.

Paroxetine e boetse e sebelisoa ho phekola maemo a mang a bophelo ba kelello a kang obsessive-compulsive disorder(OCD), panic disorder, social depression disorder, le post-traumatic stress disorder (PTSD) .Mokhoa oa eona oa ho sebetsa maemong ana o tšoana le oa oona. Ka ho eketsa maemo a serotonin bokong, Paroxetine e thusa ho fokotsa matšoao a amanang le mathata ana.


245pak

Tšebeliso ea Paroxetine e kenyelletsa maemo a mangata a bophelo bo botle ba kelello, e leng se etsang hore e be meriana e fapaneng le ea bohlokoa. Joaloka antidepressant, Paroxetine e sebelisetsoa ho kokobetsa matšoao a bothata bo boholo ba ho tepella maikutlong, ho akarelletsa le ho hlonama ho sa feleng, ho lahleheloa ke thahasello mesebetsing e tloaelehileng Ha ho phekoloa mafu a ho tšoenyeha, Paroxetine e sebetsa hantle ho fokotsa matšoao a ho tšoenyeha ka kakaretso, matšoenyeho a sechaba le mathata a ho tšoha. , le litlhaselo tsa ho tšoha, tse lumellang batho ka bomong hore ba boele ba laole maikutlo a bona le ts'ebetso ea bona ea letsatsi le letsatsi.


Ho bakuli ba nang le OCD, Paroxetine e bapala karolo ea bohlokoa ho laola maikutlo le likhothaletso tse sitisang bophelo ba bona ba letsatsi le letsatsi. Ho feta moo, Paroxetine e boetse e sebelisoa kalafong ea PTSD, moo e thusang ho fokotsa matšoao a sithabetsang a amanang le liketsahalo tse sithabetsang, joalo ka menahano e makatsang, litoro tse tšosang, ho falimeha ho feteletseng le boitšoaro ba ho qoba. tsamaisong ea maemo a mang a kang premenstrual dysphoric disorder(PMDD), matšoao a vasomotor a amanang le ho khaotsa ho ilela khoeli, le mefuta e fapa-fapaneng ea matšoao a bohloko.

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